SCHEMBL28073692

SCHEMBL28073692

COc1cnc(C(F)(F)F)nc1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 8/20 0.38
PDE4A P27815 3/20 0.36
PDE4C Q08493 3/20 0.36
PDE4D Q08499 3/20 0.36
PDE3B Q13370 3/20 0.36
PDE11A Q9HCR9 3/20 0.36
TSHR P16473 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
AURKA O14965 2/20 0.33
KDR P35968 2/20 0.33
AURKB Q96GD4 2/20 0.33
KDM4E B2RXH2 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TKT P29401 1/20 0.33
FOS P01100 2/20 0.32
JUN P05412 2/20 0.32
NFKB1 P19838 2/20 0.32
NFKB2 Q00653 2/20 0.32
RELA Q04206 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5736850 0.79 PDE4B (0.40) PDE4BPDE4APDE4CPDE4DPDE3B
SCHEMBL5736940 0.79 PDE4B (0.41) PDE4BPDE4APDE4CPDE4DPDE3B
SCHEMBL2352572 0.78 FOS (0.36) PDE4BPDE4APDE4CPDE4DPDE3B
SCHEMBL19302652 0.75 SORT1 (0.35) KDM4EALDH1A1TKTFOSJUN
SCHEMBL24975433 0.74 HTT (0.51) SMN1; SMN2L3MBTL1
SCHEMBL31292125 0.74 KDM4E (0.42) PDE4BTSHRSMN1; SMN2KDM4EL3MBTL1
Ammonia Solution, Strong SCHEMBL17353626 0.74 SORT1 (0.35) ALDH1A1TKTFOSJUNNFKB1
SCHEMBL25164042 0.73 HPGD (0.36) PDE4BPDE4APDE4CPDE4DPDE3B
SCHEMBL24975430 0.73 MKNK2 (0.40) TKT
SCHEMBL31292151 0.73 KDM4E (0.38) PDE4BPDE4APDE4CPDE4DPDE3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104254525-B aromatic ring compound TAKEDA PHARMACEUTICAL CO.,LTD. (JP) 2016-05-25 CN disclosed