SCHEMBL28074599

SCHEMBL28074599

COc1cc(-c2ccc(C(F)(F)F)cn2)ncn1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
NPSR1 Q6W5P4 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPK1 P28482 1/20 0.38
KDR P35968 1/20 0.38
MAPK14 Q16539 1/20 0.38
TNNI3K Q59H18 1/20 0.38
IDO1 P14902 1/20 0.38
TDO2 P48775 1/20 0.38
SORT1 Q99523 1/20 0.38
TRPV1 Q8NER1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL132252 0.81 GABRA1 (0.46) TSHRSMN1; SMN2NPSR1KDM4EIDO1
SCHEMBL17664492 0.77 FEN1 (0.46) KDRMAPK14TNNI3KIDO1
SCHEMBL18224103 0.76 NPSR1 (0.40) NPSR1KDM4E
SCHEMBL811160 0.76 NPSR1 (0.53) TSHRSMN1; SMN2NPSR1KDM4E
SCHEMBL29595709 0.76 NPSR1 (0.53) TSHRSMN1; SMN2NPSR1KDM4E
SCHEMBL22256396 0.75 KDM4E (0.50) TSHRSMN1; SMN2KDM4EMAPK1TRPV1
SCHEMBL706407 0.75 TSHR (0.63) TSHRSMN1; SMN2NPSR1KDM4EMAPK1
SCHEMBL30980818 0.75 TSHR (0.63) TSHRSMN1; SMN2NPSR1KDM4EMAPK1
SCHEMBL16647601 0.74 TRPA1 (0.40) NPSR1KDM4EMAPK1
SCHEMBL16635112 0.74 TRPA1 (0.42) NPSR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105612153-A Substituted sulfonamide compounds as TRPA1 conditioner HOFFMANN LA ROCHE 2016-05-25 CN disclosed