SCHEMBL28076702

SCHEMBL28076702

COc1cc(N)c(CC2CCN(CCC(O)c3ccccc3)CC2)cc1C(N)=O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.49
SLC6A4 P31645 4/20 0.48
SLC6A3 Q01959 4/20 0.48
SLC6A2 P23975 3/20 0.48
ADRA1D P25100 2/20 0.48
ADRA1A P35348 2/20 0.48
ADRA1B P35368 2/20 0.48
GRIN2D O15399 1/20 0.48
GRIN3B O60391 1/20 0.48
GRIN1 Q05586 1/20 0.48
GRIN2A Q12879 1/20 0.48
GRIN2B Q13224 1/20 0.48
GRIN2C Q14957 1/20 0.48
GRIN3A Q8TCU5 1/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
HTR1A P08908 1/20 0.47
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
DRD2 P14416 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27997741 0.92 HTR4 (0.42) ADRA1DADRA1AADRA1BGRIN2DGRIN3B
SCHEMBL28956404 0.91 SLC6A2 (0.47) SLC6A4SLC6A3SLC6A2ADRA1DADRA1A
SCHEMBL27997728 0.91 HTR4 (0.46) ADRA1DADRA1AADRA1BGRIN2DGRIN3B
SCHEMBL27997533 0.91 SLC6A2 (0.47) SLC6A4SLC6A3SLC6A2ADRA1DADRA1A
SCHEMBL27997525 0.91 MEN1 (0.43) SLC6A4ADRA1DADRA1AADRA1BMEN1
SCHEMBL27997721 0.91 ADRA1D (0.53) ADRA1DADRA1AADRA1BMEN1KMT2A
SCHEMBL27997528 0.91 HTR4 (0.42) MEN1KMT2AALDH1A1DRD2DRD4
SCHEMBL27997732 0.91 SLC6A4 (0.41) MCHR1SLC6A4SLC6A3SLC6A2GRIN2B
SCHEMBL28816405 0.88 ACHE (0.45) MEN1KMT2AALDH1A1DRD2DRD4
SCHEMBL27997523 0.88 HTR4 (0.45) MEN1KMT2AALDH1A1ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103980184-B Piperidine compounds, medical composition and its use containing this compound 爱思开生物制药株式会社 2016-08-24 CN claimed
CN-105646331-B Piperidine compounds, the medical composition and its use containing the compound 爱思开生物制药株式会社 2018-07-03 CN disclosed
CN-103980184-B Piperidine compounds, medical composition and its use containing this compound 爱思开生物制药株式会社 2016-08-24 CN disclosed