SCHEMBL2807671

SCHEMBL2807671

C#Cc1cc(C)c(N)c(C)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
TDP1 Q9NUW8 2/20 0.50
CYP3A4 P08684 2/20 0.50
TSHR P16473 2/20 0.50
TP53 P04637 1/20 0.50
POLB P06746 1/20 0.42
CYP1A1 P04798 1/20 0.33
CYP1B1 Q16678 1/20 0.33
HDAC8 Q9BY41 1/20 0.32
MAPK1 P28482 1/20 0.32
SLC6A2 P23975 1/20 0.32
GRM5 P41594 1/20 0.32
KDM4E B2RXH2 2/20 0.31
LMNA P02545 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PTPN1 P18031 1/20 0.30
PTPN6 P29350 1/20 0.30
PTPN11 Q06124 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31116962 0.84 ALDH1A1 (0.36) ALDH1A1TDP1CYP3A4TSHRTP53
SCHEMBL2806688 0.76 PTPN1 (0.35) CYP1A1CYP1B1HDAC8PTPN1PTPN6
SCHEMBL2814698 0.74 CYP1A1 (0.33) CYP1A1CYP1B1HDAC8
SCHEMBL2807287 0.74 CA1 (0.50) ALDH1A1CYP3A4CYP1A1CYP1B1KDM4E
SCHEMBL1182463 0.74 ALDH1A1 (0.50) ALDH1A1TDP1CYP3A4TSHRTP53
Methylamine SCHEMBL29029240 0.74 CYP1A1 (0.40) CYP1A1CYP1B1HDAC8GRM5
SCHEMBL3704142 0.73 ALDH1A1 (0.34) ALDH1A1TDP1CYP3A4TSHRTP53
SCHEMBL30362289 0.73 CYP3A4 (0.50) ALDH1A1TDP1CYP3A4TSHRTP53
SCHEMBL2810033 0.73 CYP3A4 (0.50) ALDH1A1TDP1CYP3A4TSHRTP53
SCHEMBL30464787 0.72 ALDH1A1 (0.48) ALDH1A1TDP1CYP3A4TSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113024583-A Preparation and application of compound containing biporphyrin 中南大学 2021-06-25 CN disclosed
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF FUJIFILM CORPORATION (JP) 2010-11-11 US disclosed
US-20100240908-A1 ACETYLENE COMPOUND FUJIFILM CORPORATION (JP) 2010-09-23 US disclosed
EP-2202221-A1 ACETYLENE COMPOUND Fujifilm Corporation (JP) 2010-06-30 EP disclosed
EP-2202220-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF Fujifilm Corporation (JP) 2010-06-30 EP disclosed
US-20100079705-A1 SUBSTRATE FOR LIQUID CRYSTAL DISPLAY DEVICE FUJIFILM CORPORATION (JP) 2010-04-01 US disclosed
US-20100079705-A1 SUBSTRATE FOR LIQUID CRYSTAL DISPLAY DEVICE FUJIFILM CORPORATION (JP) 2010-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240908-A1 ACETYLENE COMPOUND NAT1, KATNA1, KAT2B ALDH1A1 401/4885TDP1 4533/4885CYP3A4 1909/4885
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF KAT8, HDAC10, SSRP1 ALDH1A1 1480/4885TDP1 4001/4885CYP3A4 3918/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.