SCHEMBL2810033

SCHEMBL2810033

C#Cc1ccc(N)c(C)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.50
TDP1 Q9NUW8 7/20 0.50
ALDH1A1 P00352 4/20 0.50
TSHR P16473 3/20 0.50
S100B P04271 1/20 0.39
MAPK1 P28482 2/20 0.39
TP53 P04637 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
SKP2 Q13309 1/20 0.38
THRB P10828 2/20 0.37
ALOX15 P16050 2/20 0.37
RECQL P46063 1/20 0.37
HIF1A Q16665 1/20 0.37
ESR1 P03372 1/20 0.35
AR P10275 1/20 0.35
ESR2 Q92731 1/20 0.35
CASP1 P29466 1/20 0.34
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30362289 1.00 CYP3A4 (0.50) CYP3A4TDP1ALDH1A1TSHRS100B
SCHEMBL1467057 0.82 TDP1 (0.50) CYP3A4TDP1ALDH1A1TSHRMAPK1
SCHEMBL31338515 0.78 NR4A1 (0.44) CYP3A4TDP1ALDH1A1TSHRTP53
SCHEMBL4169804 0.78 NR4A1 (0.44) CYP3A4TDP1ALDH1A1TSHRTP53
SCHEMBL5718769 0.78 ALDH1A1 (0.40) TDP1ALDH1A1TSHRCA12CA1
SCHEMBL627108 0.77 CYP3A4 (0.50) CYP3A4TDP1ALDH1A1TSHRS100B
SCHEMBL10944967 0.77 CYP3A4 (0.50) CYP3A4TDP1ALDH1A1TSHRS100B
SCHEMBL3150263 0.77 ESR1 (0.38) CYP3A4TDP1ALDH1A1TSHRSMN1; SMN2
Hydrochloric Acid SCHEMBL18493517 0.76 NR4A1 (0.42) CYP3A4TDP1ALDH1A1TSHRTP53
SCHEMBL3841101 0.74 HDAC8 (0.34) CA12CA1CA2CA9CA14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9890327-B2 Phosphorescent transition metal complex, its preparation and use CITY UNIVERSITY OF HONG KONG (HK) 2018-02-13 US disclosed
US-20170114275-A1 PHOSPHORESCENT TRANSITION METAL COMPLEX, ITS PREPARATION AND USE CITY UNIVERSITY OF HONG KONG (HK) 2017-04-27 US disclosed
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF FUJIFILM CORPORATION (JP) 2010-11-11 US disclosed
CN-101868444-A Acetylenic compound, salt thereof, condensate thereof, and composition thereof FUJIFILM CORP 2010-10-20 CN disclosed
US-20100240908-A1 ACETYLENE COMPOUND FUJIFILM CORPORATION (JP) 2010-09-23 US disclosed
CN-101835752-A Heterocyclic amides useful for the treatment of cancer and psoriasis ASTRAZENECA AB 2010-09-15 CN disclosed
CN-101808982-A Acetylene compound FUJIFILM CORP 2010-08-18 CN disclosed
EP-2202221-A1 ACETYLENE COMPOUND Fujifilm Corporation (JP) 2010-06-30 EP disclosed
EP-2202220-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF Fujifilm Corporation (JP) 2010-06-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240908-A1 ACETYLENE COMPOUND NAT1, KATNA1, KAT2B CYP3A4 1909/4885TDP1 4533/4885ALDH1A1 401/4885
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF KAT8, HDAC10, SSRP1 CYP3A4 3918/4885TDP1 4001/4885ALDH1A1 1480/4885
US-20170114275-A1 PHOSPHORESCENT TRANSITION METAL COMPLEX, ITS PREPARATION AND USE DNAJA3, HSPE1, MDH2 CYP3A4 3471/4885TDP1 2894/4885ALDH1A1 3496/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.