SCHEMBL28076773

SCHEMBL28076773

COc1ccc(CC2CCN(OC(C)c3ccc(C#N)cc3)CC2)c(N)c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GPR6 P46095 3/20 0.38
ABCB1 P08183 1/20 0.38
ABCC1 P33527 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
RYR2 Q92736 1/20 0.37
HRH3 Q9Y5N1 5/20 0.36
SIGMAR1 Q99720 1/20 0.36
HTR1A P08908 3/20 0.36
SLC6A4 P31645 3/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
KDM1A O60341 1/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35
PDE10A Q9Y233 1/20 0.35
CCR6 P51684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28076593 0.87 HTR1A (0.45) GPR6RYR2HTR1ASLC6A4
SCHEMBL28076775 0.81 HTR1A (0.43) GPR6RYR2HTR1ASLC6A4
SCHEMBL28076638 0.77 HTR1A (0.46) RYR2HTR1ASLC6A4
SCHEMBL28076772 0.75 HTR1A (0.43) GPR6HTR1ASLC6A4
SCHEMBL3577962 0.74 RYR2 (0.49) RYR2SIGMAR1HTR1ASLC6A4
SCHEMBL30323089 0.72 GPR6 (0.59) GPR6HTR1ASLC6A4
SCHEMBL20524624 0.72 GPR6 (0.59) GPR6HTR1ASLC6A4
SCHEMBL3586208 0.71 MEN1 (0.43) RYR2HTR1ASLC6A4
SCHEMBL3587135 0.70 PIK3CG (0.52) RYR2HTR1ASLC6A4
SCHEMBL3574540 0.70 MTNR1A (0.44) RYR2HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103980184-B Piperidine compounds, medical composition and its use containing this compound 爱思开生物制药株式会社 2016-08-24 CN disclosed