SCHEMBL28079313

SCHEMBL28079313

O=C(O)c1ccc(CCI)nc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P4HA1 P13674 3/20 0.52
P4HTM Q9NXG6 2/20 0.52
ALDH1A1 P00352 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C9 P11712 1/20 0.52
HPGD P15428 1/20 0.52
CYP2C19 P33261 1/20 0.52
HSD17B10 Q99714 1/20 0.52
MIF P14174 1/20 0.50
GABRP O00591 1/20 0.48
GABRD O14764 1/20 0.48
GABRA1 P14867 1/20 0.48
GABRB1 P18505 1/20 0.48
GABRG2 P18507 1/20 0.48
GABRB3 P28472 1/20 0.48
GABRA5 P31644 1/20 0.48
GABRA3 P34903 1/20 0.48
GABRA2 P47869 1/20 0.48
GABRB2 P47870 1/20 0.48
GABRA4 P48169 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL152571 0.83 P4HA1 (0.53) P4HA1P4HTMALDH1A1CYP1A2CYP2C9
SCHEMBL27191301 0.81 P4HA1 (0.52) P4HA1P4HTMALDH1A1CYP1A2CYP2C9
SCHEMBL21787687 0.81 P4HA1 (0.57) P4HA1P4HTMALDH1A1CYP1A2CYP2C9
SCHEMBL565981 0.81 HCAR3 (0.58) P4HA1P4HTMALDH1A1CYP1A2CYP2C9
SCHEMBL27738856 0.81 NAPRT (0.53) P4HA1P4HTMALDH1A1CYP1A2CYP2C9
SCHEMBL28664825 0.81 GABRP (0.53) P4HA1P4HTMALDH1A1CYP1A2CYP2C9
Hydrochloric Acid SCHEMBL18740159 0.80 GABRP (0.52) P4HA1P4HTMALDH1A1CYP1A2CYP2C9
SCHEMBL20046092 0.80 P4HA1 (0.50) P4HA1P4HTMALDH1A1CYP1A2CYP2C9
SCHEMBL20423258 0.79 P4HA1 (0.48) P4HA1P4HTMALDH1A1CYP1A2CYP2C9
SCHEMBL10663641 0.79 HCAR3 (0.56) P4HA1P4HTMALDH1A1CYP1A2MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103420977-B There is the acetylene-derivative of anti-tumor activity 上海医药集团股份有限公司 2016-06-22 CN disclosed