SCHEMBL28079765

SCHEMBL28079765

Clc1ncncc1-c1ccc(Br)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
LMNA P02545 1/20 0.49
TOP2A P11388 1/20 0.43
TOP2B Q02880 1/20 0.43
DGAT1 O75907 2/20 0.38
GAA P10253 2/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
CYP1A2 P05177 4/20 0.36
CYP3A4 P08684 4/20 0.36
CYP2C19 P33261 4/20 0.36
CYP2D6 P10635 3/20 0.36
MAPK1 P28482 3/20 0.36
TP53 P04637 1/20 0.36
CYP2C9 P11712 1/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
GCGR P47871 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27399146 0.81 ALDH1A1 (0.49) MAPTSMN1; SMN2LMNADGAT1CYP1A2
SCHEMBL7013819 0.81 DGAT1 (0.41) LMNATOP2ATOP2BDGAT1CYP1A2
SCHEMBL31392405 0.80 ATM (0.46) CYP1A2CYP3A4CYP2C19CYP2D6MAPK1
SCHEMBL9046762 0.74 MEN1 (0.68) MAPTLMNAGAACYP1A2CYP3A4
SCHEMBL15023022 0.73 MAPK9 (0.59) SMN1; SMN2LMNATOP2ATOP2BKMT2A
SCHEMBL999683 0.71 MAPT (0.50) MAPTSMN1; SMN2LMNADGAT1GAA
SCHEMBL9140635 0.69 CDC25B (0.33) CDC25B
SCHEMBL28209270 0.68 ATM (0.46) MAPTSMN1; SMN2GAAMAPK1TP53
SCHEMBL29460951 0.68
SCHEMBL1344036 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104311492-B The preparation method that a kind of ACT-064992 intermediate is new 成都克莱蒙医药科技有限公司 2016-08-24 CN disclosed