SCHEMBL28080223

SCHEMBL28080223

O=C(O)CN1CCNCC1.c1cnc(N2CCCCC2)nc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.54
KDM4E B2RXH2 7/20 0.54
TDP1 Q9NUW8 3/20 0.54
SMN1; SMN2 Q16637 3/20 0.48
MDM2 Q00987 2/20 0.46
TSHR P16473 2/20 0.44
HTT P42858 1/20 0.44
CYP2D6 P10635 2/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C19 P33261 1/20 0.43
CYP1A2 P05177 1/20 0.43
HSD17B10 Q99714 1/20 0.43
USP2 O75604 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HTR1A P08908 1/20 0.42
TP53 P04637 1/20 0.41
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28223075 0.82 ALDH1A1 (0.59) ALDH1A1KDM4ETDP1SMN1; SMN2TSHR
SCHEMBL7356339 0.82 ALDH1A1 (0.66) ALDH1A1KDM4ETDP1SMN1; SMN2MDM2
Hydrochloric Acid SCHEMBL1371732 0.81 ALDH1A1 (0.64) ALDH1A1KDM4ETDP1SMN1; SMN2MDM2
2-Piperazin-1-Yl-Pyrimidine SCHEMBL10876592 0.81 KDM4E (0.70) ALDH1A1KDM4ETDP1MDM2TSHR
Piperazine SCHEMBL28070940 0.78 ALDH1A1 (0.70) ALDH1A1KDM4ETDP1SMN1; SMN2TSHR
SCHEMBL28112388 0.77 ALDH1A1 (0.51) ALDH1A1KDM4ETDP1SMN1; SMN2TSHR
Piperazine SCHEMBL28080084 0.77 ALDH1A1 (0.68) ALDH1A1KDM4ETDP1SMN1; SMN2TSHR
SCHEMBL9232046 0.75 CHRM5 (0.50) ALDH1A1SMN1; SMN2CYP1A2HSD17B10
SCHEMBL337070 0.74 HSD17B10 (0.52) SMN1; SMN2HSD17B10
SCHEMBL62990 0.74 HSD17B10 (0.52) SMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814048-B Fused tricyclic benzimidizole derivatives as TNF active regulators UCB生物制药私人有限公司 2018-03-27 CN disclosed
CN-105814048-A Fused tricyclic imidazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed