SCHEMBL28080860

SCHEMBL28080860

CC(C)c1n[nH]cc1-c1cccnc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 6/20 0.44
CYP3A4 P08684 5/20 0.44
ALDH1A1 P00352 3/20 0.44
CYP1A2 P05177 2/20 0.44
DYRK1A Q13627 3/20 0.43
GSK3B P49841 1/20 0.43
CYP2C9 P11712 4/20 0.41
CYP2C19 P33261 3/20 0.41
CYP2E1 P05181 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2B6 P20813 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
ALK Q9UM73 1/20 0.41
METAP2 P50579 1/20 0.40
SIRT3 Q9NTG7 1/20 0.40
CLK1 P49759 1/20 0.40
PDE10A Q9Y233 1/20 0.40
TDO2 P48775 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22667105 0.81 GCGR (0.38) ALDH1A1DYRK1AGSK3BADRA2AADRA2B
SCHEMBL28831872 0.80 DYRK1A (0.38) CYP3A4DYRK1AGSK3BCYP2D6ADRA2A
SCHEMBL1924022 0.76 CYP2A6 (0.50) CYP2A6CYP3A4ALDH1A1CYP1A2DYRK1A
SCHEMBL15723977 0.76 CYP2A6 (0.52) CYP2A6CYP3A4ALDH1A1CYP1A2CYP2C9
SCHEMBL4789914 0.75 CYP2A6 (0.48) CYP2A6CYP3A4ALDH1A1CYP1A2DYRK1A
SCHEMBL16051028 0.73
SCHEMBL23329265 0.72 MKNK1 (0.49) CYP2A6CYP3A4ALDH1A1CYP1A2DYRK1A
SCHEMBL2694498 0.72 NUDT1 (0.47) DYRK1AALKCLK1NUDT1
SCHEMBL30384675 0.71 METAP2 (0.47) CYP2A6CYP3A4ALDH1A1CYP1A2DYRK1A
SCHEMBL21540038 0.71 NUDT1 (0.45) CYP2A6CYP3A4ALDH1A1CYP1A2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104710420-B Azabicyclic formula compound or its salt, containing its medicine, compositions and application 大鹏药品工业株式会社 2016-07-27 CN disclosed