SCHEMBL28080906

SCHEMBL28080906

COc1ccc(CN2C(=O)C(c3ccccc3)=C(c3ccccc3)C2=O)cc1

nearest known ligand 0.71

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 3/20 0.71
NR1H3 Q13133 3/20 0.71
CASP3 P42574 2/20 0.62
CMA1 P23946 1/20 0.60
KDM4E B2RXH2 1/20 0.57
GSK3A P49840 1/20 0.57
GSK3B P49841 1/20 0.57
EP300 Q09472 1/20 0.53
MEN1 O00255 1/20 0.53
APAF1 O14727 1/20 0.53
GAA P10253 1/20 0.53
KMT2A Q03164 1/20 0.53
SENP8 Q96LD8 1/20 0.53
SENP7 Q9BQF6 1/20 0.53
SENP6 Q9GZR1 1/20 0.53
SIGMAR1 Q99720 1/20 0.51
CHRM5 P08912 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30320663 0.94 NR1H2 (0.71) NR1H2NR1H3CASP3CMA1KDM4E
SCHEMBL28169955 0.89 NR1H2 (0.62) NR1H2NR1H3CASP3CMA1KDM4E
SCHEMBL4450601 0.84 NR1H2 (1.00) NR1H2NR1H3CASP3GSK3BEP300
SCHEMBL15437828 0.83 NR1H2 (0.70) NR1H2NR1H3CASP3CMA1GSK3A
SCHEMBL45154 0.82 CASP3 (0.88) CASP3CMA1KDM4EMEN1APAF1
SCHEMBL30296449 0.82 CASP3 (0.88) CASP3CMA1KDM4EMEN1APAF1
SCHEMBL28080973 0.82 NR1H2 (0.54) NR1H2NR1H3KDM4EMEN1KMT2A
SCHEMBL28080839 0.80 NR1H2 (0.68) NR1H2NR1H3CASP3CMA1MEN1
SCHEMBL4693569 0.80 NR1H2 (0.81) NR1H2NR1H3CASP3GSK3BL3MBTL1
SCHEMBL4692898 0.80 NR1H2 (0.81) NR1H2NR1H3CASP3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103804108-B A kind of method preparing primary amine 沈阳药科大学 2016-08-03 CN disclosed