SCHEMBL28082066

SCHEMBL28082066

COC(=O)C(C)Oc1c(F)cc(F)cc1[N+](=O)[O-]

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.42
ALDH1A1 P00352 4/20 0.40
HSPB1 P04792 1/20 0.38
ATM Q13315 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
SRD5A2 P31213 1/20 0.37
MEN1 O00255 2/20 0.36
TTR P02766 2/20 0.36
TPMT P51580 1/20 0.36
ABCB1 P08183 1/20 0.35
ABCC1 P33527 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30806393 1.00 KMT2A (0.42) KMT2AALDH1A1HSPB1ATMTDP1
SCHEMBL28082067 1.00 KMT2A (0.42) KMT2AALDH1A1HSPB1ATMTDP1
SCHEMBL30806384 1.00 KMT2A (0.42) KMT2AALDH1A1HSPB1ATMTDP1
SCHEMBL28529013 0.87 ALDH1A1 (0.38) KMT2AALDH1A1SRD5A2MEN1TPMT
SCHEMBL28533883 0.87 ALDH1A1 (0.38) KMT2AALDH1A1SRD5A2MEN1TTR
SCHEMBL18305024 0.87 ALDH1A1 (0.38) KMT2AALDH1A1SRD5A2MEN1TTR
SCHEMBL18304994 0.87 ALDH1A1 (0.38) KMT2AALDH1A1SRD5A2MEN1TPMT
SCHEMBL28082061 0.87 MAPT (0.42) KMT2AALDH1A1HSPB1ATMTDP1
SCHEMBL28082062 0.87 MAPT (0.42) KMT2AALDH1A1HSPB1ATMTDP1
SCHEMBL18128032 0.86 SRD5A2 (0.41) KMT2AALDH1A1HSPB1ATMTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814054-A Fused imidazole and pyrazole derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed