SCHEMBL28084402

SCHEMBL28084402

Cc1cc(C)cc(NC(=O)c2ccccc2I)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.67
KMT2A Q03164 4/20 0.67
TDP1 Q9NUW8 1/20 0.67
POLB P06746 1/20 0.60
THRB P10828 2/20 0.56
ALDH1A1 P00352 3/20 0.53
PKM P14618 1/20 0.53
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
P2RX1 P51575 1/20 0.51
TMPRSS4 Q9NRS4 1/20 0.51
MAPT P10636 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
HPGD P15428 2/20 0.50
KDM4E B2RXH2 1/20 0.50
RXFP1 Q9HBX9 1/20 0.50
RAB9A P51151 2/20 0.49
NPC1 O15118 1/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17376723 0.87 MEN1 (0.70) MEN1KMT2ATDP1POLBALDH1A1
SCHEMBL11590379 0.85 KMT2A (0.74) MEN1KMT2ATDP1POLBALDH1A1
SCHEMBL30030085 0.85 KMT2A (0.74) MEN1KMT2ATDP1POLBALDH1A1
SCHEMBL1961258 0.81 FADS1 (0.69) MEN1KMT2APOLBTHRBALDH1A1
Benodanil SCHEMBL18736 0.80 MEN1 (1.00) MEN1KMT2ATDP1POLBALDH1A1
Benodanil SCHEMBL29402073 0.80 MEN1 (1.00) MEN1KMT2ATDP1POLBALDH1A1
SCHEMBL28608407 0.80 RAB9A (0.68) MEN1KMT2APOLBP2RX1TMPRSS4
SCHEMBL1496329 0.80 MEN1 (0.60) MEN1KMT2ATDP1POLBTHRB
SCHEMBL6811221 0.78 MEN1 (0.74) MEN1KMT2ATDP1POLBALDH1A1
SCHEMBL28493350 0.78 ALDH1A1 (0.68) MEN1KMT2ATDP1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104163799-B 3-amino-4-Cyanoisoquinoline-1(2H) preparation method of-one derivant 苏州大学 2016-08-17 CN disclosed