Hexobendine

Hexobendine

SCHEMBL28086121

CCOC(=O)COc1ccc2c(C)c(CCN(CC)CC)c(=O)oc2c1.COc1cc(C(=O)OCCCN(C)CCN(C)CCCOC(=O)c2cc(OC)c(OC)c(OC)c2)cc(OC)c1OC

nearest known ligand 0.50

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.50
ALDH1A1 P00352 7/20 0.50
HPGD P15428 7/20 0.50
HSD17B10 Q99714 5/20 0.50
SCN1A P35498 1/20 0.49
SCN2A Q99250 1/20 0.49
SCN3A Q9NY46 1/20 0.49
CA12 O43570 8/20 0.48
CA9 Q16790 8/20 0.48
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KMT2A Q03164 3/20 0.46
TSHR P16473 1/20 0.46
MEN1 O00255 2/20 0.45
ATM Q13315 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
THPO P40225 1/20 0.45
MTOR P42345 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chromonar SCHEMBL29724124 0.82 KDM4E (0.67) KDM4EALDH1A1HPGDHSD17B10CA12
Chromonar SCHEMBL309094 0.82 KDM4E (0.67) KDM4EALDH1A1HPGDHSD17B10CA12
SCHEMBL4395187 0.82 KDM4E (0.65) KDM4EALDH1A1HPGDHSD17B10CA12
Chromonar SCHEMBL122836 0.82 KDM4E (0.66) KDM4EALDH1A1HPGDHSD17B10CA12
Chromonar SCHEMBL29351852 0.82 KDM4E (0.66) KDM4EALDH1A1HPGDHSD17B10CA12
SCHEMBL29944843 0.72 KDM4E (0.55) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL7141692 0.72 KDM4E (0.55) KDM4EALDH1A1HPGDHSD17B10NPC1
Hexobendine SCHEMBL125629 0.70 SCN1A (1.00) SCN1ASCN2ASCN3ASMN1; SMN2KMT2A
SCHEMBL18095433 0.70 ALDH1A1 (0.70) KDM4EALDH1A1HPGDHSD17B10CA12
Chromonar SCHEMBL28142053 0.69 THRA (0.53) KDM4EALDH1A1HPGDHSD17B10SCN1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103717597-B Heterocyclic compounds as kinase inhibitors 原真股份有限公司 2017-07-04 CN disclosed
CN-103492389-B Pyrazolo [4,3-d] pyrimidine as inhibitors of kinases 原真股份有限公司 2016-09-14 CN disclosed