Fenpiverinium

Fenpiverinium

SCHEMBL28086315

CN(C)CCC=O.C[N+]1(CCC(C(N)=O)(c2ccccc2)c2ccccc2)CCCCC1

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.43
DRD3 P35462 2/20 0.43
DRD2 P14416 1/20 0.43
CHRM3 P20309 10/20 0.43
CHRM2 P08172 6/20 0.43
CHRM1 P11229 2/20 0.43
CHRM4 P08173 1/20 0.43
CHRM5 P08912 1/20 0.43
DRD4 P21917 1/20 0.41
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.39
KCNH2 Q12809 2/20 0.38
LMNA P02545 1/20 0.38
CYP2D6 P10635 1/20 0.38
KDM4E B2RXH2 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
SLC22A2 O15244 1/20 0.35
SLC22A1 O15245 1/20 0.35
PGR P06401 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fenpiverinium SCHEMBL1650132 0.86 CHRM3 (0.55) OPRM1DRD3DRD2CHRM3CHRM2
Buzepide SCHEMBL3498775 0.85 CHRM3 (0.57) CHRM3CHRM2CHRM1CHRM4CHRM5
Fenpiverinium SCHEMBL23654 0.85 CHRM3 (0.53) CHRM3CHRM2CHRM1CHRM4CHRM5
Iodide SCHEMBL29558329 0.66 CHRM2 (0.83) OPRM1DRD3DRD2CHRM3CHRM2
SCHEMBL9295790 0.63 CHRM3 (0.59) OPRM1DRD3DRD2CHRM3CHRM2
SCHEMBL3900689 0.63 OPRM1 (0.58) OPRM1DRD3DRD2CHRM3CHRM2
SCHEMBL9426731 0.62 OPRM1 (0.54) OPRM1DRD3DRD2CHRM3CHRM2
Normethadone SCHEMBL24337 0.62 OPRM1 (1.00) OPRM1DRD3DRD2CHRM3CHRM2
Benzene SCHEMBL9326315 0.62 HRH1 (0.39) OPRM1DRD3DRD2CHRM3CHRM2
SCHEMBL13541547 0.62 KCNH2 (0.74) OPRM1DRD3DRD2CHRM3CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103717597-B Heterocyclic compounds as kinase inhibitors 原真股份有限公司 2017-07-04 CN disclosed
CN-103492389-B Pyrazolo [4,3-d] pyrimidine as inhibitors of kinases 原真股份有限公司 2016-09-14 CN disclosed