SCHEMBL2808633

SCHEMBL2808633

Nc1cccc(C#Cc2ccc3ccccc3n2)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 3/20 0.55
GRM5 P41594 5/20 0.51
KCNH2 Q12809 3/20 0.51
PIK3CA P42336 1/20 0.50
MTOR P42345 1/20 0.50
PDK1 Q15118 1/20 0.50
HTR3A P46098 1/20 0.45
NCF1 P14598 1/20 0.42
NOS2 P35228 1/20 0.42
BACE1 P56817 1/20 0.42
GRM4 Q14833 1/20 0.41
ASIC3 Q9UHC3 1/20 0.39
RAB9A P51151 3/20 0.39
MEN1 O00255 2/20 0.39
NPC1 O15118 2/20 0.39
KMT2A Q03164 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL484570 0.82 GRM5 (0.56) TTRGRM5KCNH2PIK3CAMTOR
SCHEMBL12884290 0.82 TTR (0.62) TTRGRM5KCNH2NCF1NOS2
SCHEMBL5778843 0.81 GRM5 (0.62) TTRGRM5KCNH2NCF1NOS2
SCHEMBL2808776 0.81 TTR (0.62) TTRGRM5KCNH2RAB9AMEN1
SCHEMBL2807844 0.81 TTR (0.55) TTRGRM5KCNH2RAB9AMEN1
SCHEMBL4713149 0.81 TTR (0.55) TTRGRM5KCNH2
SCHEMBL12884286 0.79 GRM5 (0.65) TTRGRM5KCNH2NCF1NOS2
SCHEMBL4968126 0.75 CYP3A4 (0.58) PIK3CAMTORPDK1ASIC3RAB9A
SCHEMBL4711036 0.74 GRM5 (0.67) GRM5RAB9AMEN1NPC1KMT2A
SCHEMBL2811255 0.73 MAPT (0.62) KCNH2PIK3CAMTORPDK1ASIC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF FUJIFILM CORPORATION (JP) 2010-11-11 US disclosed
US-20100240908-A1 ACETYLENE COMPOUND FUJIFILM CORPORATION (JP) 2010-09-23 US disclosed
EP-2202221-A1 ACETYLENE COMPOUND Fujifilm Corporation (JP) 2010-06-30 EP disclosed
EP-2202220-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF Fujifilm Corporation (JP) 2010-06-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100240908-A1 ACETYLENE COMPOUND NAT1, KATNA1, KAT2B TTR 3597/4885GRM5 2797/4885KCNH2 382/4885
US-20100286353-A1 ACETYLENE COMPOUND, SALT THEREOF, CONDENSATE THEREOF, AND COMPOSITION THEREOF KAT8, HDAC10, SSRP1 TTR 3025/4885GRM5 3664/4885KCNH2 3430/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.