Cinepazide

Cinepazide

SCHEMBL28086342

COc1cc(/C=C/C(=O)N2CCN(CC(=O)N3CCCC3)CC2)cc(OC)c1OC.O=C(OCCN1CCCCCC1)C(c1ccsc1)C1CCCCC1

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.47
ALDH1A1 P00352 6/20 0.47
HPGD P15428 3/20 0.47
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
TRPV1 Q8NER1 1/20 0.39
KMT2A Q03164 2/20 0.39
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPT P10636 2/20 0.38
APP P05067 1/20 0.37
STAT6 P42226 1/20 0.37
TP53 P04637 1/20 0.37
HSD17B10 Q99714 1/20 0.37
BCHE P06276 3/20 0.36
ACHE P22303 3/20 0.36
MAOA P21397 2/20 0.36
MAOB P27338 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28790703 0.78 ALDH1A1 (0.73) KDM4EALDH1A1HPGDCYP3A4CYP2C19
Cinepazide SCHEMBL8839976 0.78 ALDH1A1 (0.77) KDM4EALDH1A1HPGDCYP3A4CYP2C19
Cinepazide SCHEMBL34092 0.78 ALDH1A1 (0.77) KDM4EALDH1A1HPGDCYP3A4CYP2C19
Cetiedil SCHEMBL14169136 0.76 CYP3A4 (0.44) HPGDCYP3A4KMT2ATDP1TP53
Cetiedil SCHEMBL458084 0.76 CYP3A4 (0.44) HPGDCYP3A4KMT2ATDP1TP53
Fumaric Acid SCHEMBL11710489 0.76 KDM4E (0.69) KDM4EALDH1A1HPGDCYP3A4CYP2C19
Cinepazide SCHEMBL11009911 0.76 KDM4E (0.72) KDM4EALDH1A1HPGDCYP3A4CYP2C19
Cinepazide SCHEMBL27666991 0.75 KDM4E (0.71) KDM4EALDH1A1HPGDCYP3A4CYP2C19
Cinepazide SCHEMBL1062368 0.75 KDM4E (0.71) KDM4EALDH1A1HPGDCYP3A4CYP2C19
SCHEMBL10646647 0.73 KDM4E (0.67) KDM4EALDH1A1HPGDCYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103717597-B Heterocyclic compounds as kinase inhibitors 原真股份有限公司 2017-07-04 CN disclosed
CN-103492389-B Pyrazolo [4,3-d] pyrimidine as inhibitors of kinases 原真股份有限公司 2016-09-14 CN disclosed