SCHEMBL28089157

SCHEMBL28089157

O=C(O)c1cc[c]nc1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.47
LMNA P02545 1/20 0.47
ALDH1A1 P00352 5/20 0.39
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
TSHR P16473 4/20 0.36
TP53 P04637 1/20 0.36
CASP1 P29466 1/20 0.36
ALOX15 P16050 3/20 0.36
CYP1A2 P05177 1/20 0.36
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
HSP90AA1 P07900 1/20 0.33
KDM4E B2RXH2 4/20 0.32
TDP1 Q9NUW8 2/20 0.32
NR4A1 P22736 1/20 0.32
DAO P14920 1/20 0.32
KDM5A P29375 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
MAPT P10636 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2438107 0.75 GABRP (0.46) SMN1; SMN2ALDH1A1ALOX15CYP1A2KDM4E
SCHEMBL8629182 0.71 SMN1; SMN2 (0.42) SMN1; SMN2LMNAALDH1A1KEAP1NFE2L2
SCHEMBL400674 0.67 EGFR (0.54) SMN1; SMN2LMNAALDH1A1KEAP1NFE2L2
SCHEMBL8487622 0.66 ALDH1A1 (0.47) LMNAALDH1A1KEAP1TSHRALOX15
SCHEMBL16278616 0.66 NR4A1 (0.44) SMN1; SMN2LMNAALDH1A1TSHRALOX15
Hydrochloric Acid SCHEMBL921288 0.65 EGFR (0.53) SMN1; SMN2LMNAALDH1A1KEAP1NFE2L2
SCHEMBL7444717 0.65 ALDH1A1 (0.37) SMN1; SMN2LMNAALDH1A1TSHRTP53
SCHEMBL29378242 0.65 SMN1; SMN2 (0.50) SMN1; SMN2LMNAALDH1A1KEAP1NFE2L2
SCHEMBL56617 0.65 SMN1; SMN2 (0.50) SMN1; SMN2LMNAALDH1A1KEAP1NFE2L2
SCHEMBL750508 0.64 ALDH1A1 (0.50) SMN1; SMN2LMNAALDH1A1TSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103608332-B Pyridine-2-amides useful as CB2 agonists 霍夫曼-拉罗奇有限公司 2016-09-28 CN disclosed