SCHEMBL28089176

SCHEMBL28089176

CCOn1cnc(-c2cc(OC)cc(OC)c2)c1-c1ccc(OC)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.41
PTGS1 P23219 4/20 0.41
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
MAPK1 P28482 1/20 0.38
CYP17A1 P05093 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
CALM1 P0DP23 1/20 0.36
USP2 O75604 1/20 0.36
PHF8 Q9UPP1 1/20 0.36
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
HPGD P15428 1/20 0.35
PDE7A Q13946 1/20 0.35
PDE3A Q14432 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28089178 0.95 ALDH1A1 (0.40) PTGS2PTGS1PDGFRBPDGFRAALDH1A1
SCHEMBL27934206 0.82 PHF8 (0.50) PTGS2PTGS1PDGFRBPDGFRAALDH1A1
SCHEMBL15664971 0.81 PTGS2 (0.42) PTGS2PTGS1PDGFRBPDGFRAL3MBTL1
SCHEMBL15664969 0.77 PDGFRB (0.39) PTGS2PTGS1PDGFRBPDGFRAALDH1A1
SCHEMBL28089068 0.77 PTGS2 (0.43) PTGS2PTGS1PDGFRBPDGFRAALDH1A1
SCHEMBL15664970 0.76 PTGS2 (0.42) PTGS2PDGFRBPDGFRAALDH1A1KDM4E
SCHEMBL15664996 0.76 PTGS2 (0.47) PTGS2PTGS1PDGFRBPDGFRAL3MBTL1
SCHEMBL15664763 0.71 IDO1 (0.51) PDGFRBPDGFRAALDH1A1KDM4EMAPK1
SCHEMBL27934237 0.71 PTGS2 (0.43) PTGS2ALDH1A1MAPK1L3MBTL1CALM1
SCHEMBL27934224 0.70 PHF8 (0.45) PDGFRBPDGFRAL3MBTL1PHF8SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105753787-A Tumor-targeting-medicine Combretastatin A4 derivatives 南京圣和药业股份有限公司 2016-07-13 CN disclosed