SCHEMBL28089302

SCHEMBL28089302

CC(C)(C)OC(=O)N1CCCCC1c1cccc(C(N)=O)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP14 Q460N5 3/20 0.53
PARP10 Q53GL7 1/20 0.53
RIPK1 Q13546 2/20 0.47
CFB P00751 1/20 0.46
CHEK2 O96017 1/20 0.44
NR1H2 P55055 2/20 0.43
NR1H3 Q13133 2/20 0.43
GPR119 Q8TDV5 1/20 0.43
UCHL1 P09936 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TMEM97 Q5BJF2 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
PARP1 P09874 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31226567 0.86 RIPK1 (0.49) PARP14PARP10RIPK1NR1H2NR1H3
SCHEMBL30550978 0.86 RIPK1 (0.49) PARP14PARP10RIPK1NR1H2NR1H3
SCHEMBL322073 0.86 RIPK1 (0.52) RIPK1NR1H2NR1H3UCHL1ALDH1A1
SCHEMBL31226730 0.86 RIPK1 (0.49) PARP14PARP10RIPK1NR1H2NR1H3
SCHEMBL321319 0.86 RIPK1 (0.52) RIPK1NR1H2NR1H3UCHL1ALDH1A1
SCHEMBL25320429 0.86 RIPK1 (0.49) PARP14PARP10RIPK1NR1H2NR1H3
SCHEMBL26693383 0.85 GPR119 (0.52) PARP14PARP10RIPK1CFBCHEK2
SCHEMBL21611363 0.84 RIPK1 (0.50) RIPK1NR1H2NR1H3UCHL1ALDH1A1
SCHEMBL23646533 0.84 RIPK1 (0.50) RIPK1NR1H2NR1H3UCHL1ALDH1A1
SCHEMBL8214939 0.84 ROCK2 (0.53) RIPK1NR1H2NR1H3UCHL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105849096-B Piperidine derivatives having multimodal activity against pain 埃斯蒂文制药股份有限公司 2019-11-29 CN disclosed
CN-105849096-A Piperidine derivatives having multimodal activity against pain 埃斯蒂文博士实验室股份有限公司 2016-08-10 CN disclosed