SCHEMBL28089985

SCHEMBL28089985

CNC(=O)c1cccc(C(N)=O)c1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.50
GAA P10253 2/20 0.48
CHEK1 O14757 1/20 0.41
MAP4K4 O95819 1/20 0.41
TYK2 P29597 4/20 0.41
JAK2 O60674 3/20 0.41
JAK1 P23458 3/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MTNR1A P48039 1/20 0.41
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
PARP1 P09874 1/20 0.39
METAP2 P50579 1/20 0.38
CYP2C9 P11712 1/20 0.38
BRD4 O60885 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL465699 0.85 G6PD (0.55) PLK1GAACHEK1MAP4K4KDM4E
SCHEMBL40536 0.83 ALDH1A1 (0.54) GAACHEK1MAP4K4KDM4EALDH1A1
SCHEMBL5252014 0.82 PLK1 (0.52) PLK1GAAKDM4EALDH1A1MAPT
SCHEMBL4666198 0.82 GAA (0.59) PLK1GAACHEK1MAP4K4TYK2
SCHEMBL30064209 0.82 GAA (0.59) PLK1GAACHEK1MAP4K4TYK2
SCHEMBL31038153 0.81 PLK1 (0.50) PLK1GAAKDM4EALDH1A1MAPT
SCHEMBL635088 0.81 PLK1 (0.50) PLK1GAAKDM4EALDH1A1MAPT
SCHEMBL19416407 0.81 PLK1 (0.50) PLK1GAACHEK1MAP4K4TYK2
SCHEMBL3341725 0.81 PLK1 (0.50) PLK1GAACHEK1MAP4K4TYK2
Hydrochloric Acid SCHEMBL29001816 0.80 GAA (0.57) PLK1GAACHEK1MAP4K4TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104230831-B As PI3 kinases and the triaizine compounds of mTOR inhibitors 惠氏有限责任公司 2016-08-24 CN disclosed