SCHEMBL28090366

SCHEMBL28090366

O=C(O)c1ccccc1Oc1ccc([N+](=O)[O-])c(Cl)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.55
MEN1 O00255 3/20 0.55
KMT2A Q03164 3/20 0.55
TTR P02766 2/20 0.55
PPOX P50336 1/20 0.55
HPSE Q9Y251 1/20 0.51
F10 P00742 1/20 0.50
AKR1C3 P42330 3/20 0.47
AKR1C2 P52895 3/20 0.47
AKR1C1 Q04828 2/20 0.47
AKR1B10 O60218 1/20 0.47
AKR1B1 P15121 1/20 0.47
AKR1C4 P17516 1/20 0.47
SLC25A1 P53007 1/20 0.46
MERTK Q12866 1/20 0.45
ALB P02768 1/20 0.45
THRB P10828 1/20 0.45
HPGD P15428 1/20 0.44
LMNA P02545 2/20 0.44
MAPT P10636 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10784715 0.88 TDP1 (0.58) TDP1MEN1KMT2ATTRPPOX
SCHEMBL16792618 0.85 SLC6A4 (0.51) TDP1MEN1KMT2ATTRPPOX
SCHEMBL16814217 0.85 TDP1 (0.50) TDP1MEN1KMT2ATTRPPOX
SCHEMBL80744 0.84 TDP1 (0.67) TDP1MEN1KMT2ATTRPPOX
SCHEMBL706437 0.84 HPSE (0.51) TDP1MEN1KMT2ATTRPPOX
SCHEMBL8740792 0.82 HPGD (0.51) TDP1MEN1KMT2AHPSESLC25A1
SCHEMBL4739689 0.82 KMO (0.56) ALDH1A1
SCHEMBL30775030 0.82 KMO (0.56) ALDH1A1
SCHEMBL10502108 0.80 MEN1 (0.54) MEN1KMT2AHPSEF10SLC25A1
SCHEMBL10663721 0.80 TDP1 (0.69) TDP1MEN1KMT2ATTRPPOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105793252-A Inhibitors of bruton's tyrosine kinase 豪夫迈·罗氏有限公司 2016-07-20 CN disclosed