SCHEMBL28090668

SCHEMBL28090668

O=C(c1ccccc1)c1cnn(-c2ccccc2Br)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.39
NPC1 O15118 4/20 0.39
RAB9A P51151 4/20 0.39
ALOX15 P16050 1/20 0.39
HTT P42858 1/20 0.39
HDAC1 Q13547 1/20 0.38
MAPK14 Q16539 4/20 0.37
ALDH1A1 P00352 3/20 0.37
CNR2 P34972 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.36
MEN1 O00255 2/20 0.35
AKR1C3 P42330 1/20 0.35
PKM P14618 2/20 0.35
HSP90AA1 P07900 1/20 0.35
CCR6 P51684 1/20 0.35
ATM Q13315 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
TLR9 Q9NR96 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28832952 0.82 ADORA2A (0.42) KMT2ANPC1RAB9AHTTHDAC1
SCHEMBL28090836 0.80 HDAC1 (0.51) KMT2ANPC1RAB9AHDAC1MAPK14
SCHEMBL28090835 0.79 HTT (0.47) KMT2ANPC1RAB9AALOX15HTT
SCHEMBL28090558 0.79 MAPK14 (0.38) KMT2ANPC1RAB9AHDAC1MAPK14
SCHEMBL28090536 0.76 SMN1; SMN2 (0.50) KMT2ANPC1RAB9AALOX15HTT
SCHEMBL28832969 0.75 KDM4E (0.47) KMT2AHTTHDAC1MAPK14ALDH1A1
SCHEMBL28090831 0.73 MAPK14 (0.52) KMT2ANPC1RAB9AALOX15HDAC1
SCHEMBL28090523 0.73 MAPT (0.44) KMT2ANPC1RAB9AHTTHDAC1
SCHEMBL28090559 0.70 MAPK14 (0.55) KMT2ANPC1RAB9AHTTMAPK14
SCHEMBL28090834 0.70 HDAC1 (0.49) KMT2ANPC1RAB9AHDAC1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106187923-A 2 aryl 4 aroyl triazole compounds and application thereof 沈阳药科大学 2016-12-07 CN disclosed