SCHEMBL28090536

SCHEMBL28090536

O=C(c1ccccc1)c1cnn(-c2cccc(Br)c2)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.50
HTT P42858 2/20 0.49
MAPT P10636 2/20 0.49
ALDH1A1 P00352 2/20 0.49
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HDAC1 Q13547 1/20 0.44
ALOX15 P16050 1/20 0.42
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.39
POLB P06746 1/20 0.39
MAPK14 Q16539 2/20 0.39
RPA1 P27694 1/20 0.38
BRD4 O60885 1/20 0.38
ATM Q13315 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28090836 0.85 HDAC1 (0.51) ALDH1A1MEN1KMT2AHDAC1ADORA2A
SCHEMBL28090835 0.85 HTT (0.47) HTTMAPTALDH1A1MEN1KMT2A
SCHEMBL28090518 0.77 MAPT (0.54) SMN1; SMN2HTTMAPTALDH1A1MEN1
SCHEMBL28090831 0.76 MAPK14 (0.52) MAPTALDH1A1MEN1KMT2AHDAC1
SCHEMBL28090668 0.76 KMT2A (0.39) SMN1; SMN2HTTMAPTALDH1A1MEN1
SCHEMBL28090523 0.76 MAPT (0.44) SMN1; SMN2HTTMAPTALDH1A1MEN1
SCHEMBL28090834 0.76 HDAC1 (0.49) ALDH1A1MEN1KMT2AHDAC1ADORA2A
SCHEMBL2497315 0.73 SMN1; SMN2 (0.50) SMN1; SMN2HTTMAPTALDH1A1MEN1
SCHEMBL28090559 0.73 MAPK14 (0.55) SMN1; SMN2HTTMAPTALDH1A1MEN1
SCHEMBL28278292 0.73 GABRA1 (0.45) SMN1; SMN2HTTMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106187923-A 2 aryl 4 aroyl triazole compounds and application thereof 沈阳药科大学 2016-12-07 CN disclosed