SCHEMBL28092540

SCHEMBL28092540

Brc1cncc(C2[CH]C2)c1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.36
HCAR2 Q8TDS4 1/20 0.36
CHRNB2 P17787 8/20 0.33
CHRNA4 P43681 8/20 0.33
CHRNB4 P30926 3/20 0.33
CHRNA3 P32297 3/20 0.33
CYP2A6 P11509 1/20 0.32
KDM4E B2RXH2 1/20 0.32
SMYD3 Q9H7B4 1/20 0.32
PTK2 Q05397 1/20 0.32
ALOX15 P16050 1/20 0.32
HTT P42858 1/20 0.32
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1426303 0.76 POLB (0.38) POLBHCAR2CHRNB2CHRNA4CHRNB4
SCHEMBL29845299 0.76 POLB (0.38) POLBHCAR2CHRNB2CHRNA4CHRNB4
SCHEMBL13073608 0.74 CYP2A6 (0.31) POLBHCAR2CYP2A6
SCHEMBL744158 0.72 TSHR (0.37) POLBHCAR2CHRNB2CHRNA4CHRNB4
SCHEMBL31014511 0.72 CYP11B2 (0.46) POLBHCAR2CHRNB2CHRNA4KDM4E
SCHEMBL15463774 0.71 CYP11B2 (0.36) POLBHCAR2CHRNB2CHRNA4CHRNB4
SCHEMBL30132809 0.71 CYP11B1 (0.43) POLBHCAR2CHRNB2CHRNA4CHRNB4
SCHEMBL1356433 0.71 CYP11B1 (0.43) POLBHCAR2CHRNB2CHRNA4CHRNB4
SCHEMBL20242412 0.70 CHRNB2 (0.32) POLBHCAR2CHRNB2CHRNA4CHRNB4
SCHEMBL748571 0.69 CHRNB2 (0.34) POLBHCAR2CHRNB2CHRNA4CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105849097-A Substituted pyridine derivatives as GSK-3 inhibitors 百时美施贵宝公司 2016-08-10 CN disclosed