SCHEMBL28093134

SCHEMBL28093134

c1ccc(Cc2cnc3ccc(-n4cccn4)cc3c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.41
KLKB1 P03952 2/20 0.40
KLK1 P06870 2/20 0.40
HRH3 Q9Y5N1 1/20 0.39
DRD2 P14416 1/20 0.39
DRD4 P21917 1/20 0.39
DRD3 P35462 1/20 0.39
MPO P05164 2/20 0.38
MAPK1 P28482 2/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
NOTUM Q6P988 1/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
NLRP3 Q96P20 2/20 0.37
RORC P51449 5/20 0.37
BTK Q06187 1/20 0.36
CDC7 O00311 1/20 0.36
AURKA O14965 1/20 0.36
CHUK O15111 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27565523 0.73 CYP11B1 (0.56) HRH3MAPK1KDM4EALDH1A1NOTUM
SCHEMBL28046310 0.73 NCOA3 (0.56) HRH3MAPK1KDM4EALDH1A1NOTUM
SCHEMBL3353525 0.72 EGFR (0.46) HRH3MAPK1KDM4EALDH1A1NOTUM
SCHEMBL6933468 0.72 PDGFRB (0.53) KDM4EALDH1A1
SCHEMBL22926854 0.72 PDE10A (0.49) KDM4EALDH1A1
SCHEMBL12277481 0.72 HTT (0.41) LMNAKDM4EALDH1A1
SCHEMBL12117421 0.70 CHRM1 (0.46) LMNADRD2DRD4DRD3MPO
SCHEMBL3665773 0.69 NOTUM (0.53) LMNAHRH3DRD2DRD4DRD3
SCHEMBL6779647 0.67 NOTUM (0.50) LMNAHRH3DRD2DRD4DRD3
SCHEMBL7733429 0.66 KDM4E (0.42) KLKB1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105829294-A METHYLENE LINKED QUINOLINYL MODULATORS OF ROR-GAMMA-T 詹森药业有限公司 2016-08-03 CN disclosed