SCHEMBL3353525

SCHEMBL3353525

c1cnn(-c2ccc3ncncc3c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.46
NOTUM Q6P988 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43
PIK3CD O00329 1/20 0.43
PIK3CA P42336 1/20 0.43
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPK1 P28482 1/20 0.41
LCK P06239 1/20 0.40
KIT P10721 1/20 0.40
SRC P12931 1/20 0.40
KDR P35968 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.39
NLRP3 Q96P20 2/20 0.39
FGFR4 P22455 1/20 0.38
TDO2 P48775 1/20 0.37
OPRM1 P35372 1/20 0.37
OPRL1 P41146 1/20 0.37
PDK2 Q15119 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28046310 0.80 NCOA3 (0.56) NOTUMHRH3KDM4EALDH1A1MAPK1
SCHEMBL27389898 0.78 EGFR (0.51) EGFRPIK3CDPIK3CAMKNK2NCOA3
SCHEMBL27837893 0.74 NCOA3 (0.66) EGFRNOTUMMKNK2NCOA3
SCHEMBL27565523 0.73 CYP11B1 (0.56) NOTUMHRH3KDM4EALDH1A1MAPK1
SCHEMBL27867723 0.72 NOTUM (0.41) NOTUMHRH3PIK3CDPIK3CAKDM4E
SCHEMBL28093134 0.72 LMNA (0.41) NOTUMHRH3KDM4EALDH1A1MAPK1
SCHEMBL6779647 0.72 NOTUM (0.50) NOTUMHRH3KDM4EALDH1A1MAPK1
SCHEMBL3665773 0.72 NOTUM (0.53) NOTUMHRH3KDM4EALDH1A1MAPK1
SCHEMBL3974447 0.71 HRH3 (0.53) NOTUMHRH3KDM4EALDH1A1MAPK1
SCHEMBL2241300 0.71 MAPK9 (0.58) EGFRPIK3CDPIK3CAKDRMKNK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010056758-A1 QUINAZOLINE DERIVATIVES AS KINASE INHIBITORS FENG YANGBO (US) 2010-05-20 WO disclosed