SCHEMBL28096009

SCHEMBL28096009

COc1ccc(-c2n[nH]c(-c3cc(OC)c(OC)c(OC)c3)n2)cc1OCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.51
PDE4B Q07343 1/20 0.51
PDE4C Q08493 1/20 0.51
PDE4D Q08499 1/20 0.51
ABCB1 P08183 2/20 0.48
S1PR1 P21453 1/20 0.48
NR1H2 P55055 1/20 0.47
NR1H3 Q13133 1/20 0.47
KDM4E B2RXH2 3/20 0.47
TSHR P16473 3/20 0.47
POLB P06746 1/20 0.47
HSD17B10 Q99714 2/20 0.46
MAPT P10636 3/20 0.45
MAPK1 P28482 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
USP2 O75604 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
PSEN1 P49768 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28096012 0.88 PDE4A (0.48) PDE4APDE4BPDE4CPDE4DABCB1
SCHEMBL28096083 0.83 MAPT (0.49) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL17279690 0.82 NR1H2 (0.60) NR1H2NR1H3KDM4ETSHRPOLB
Hydrochloric Acid SCHEMBL6581075 0.80 ADORA2A (0.58) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL17280055 0.79 KDM4E (0.60) S1PR1NR1H2NR1H3KDM4ETSHR
SCHEMBL15117081 0.79 NR1H2 (0.63) S1PR1NR1H2NR1H3KDM4ETSHR
SCHEMBL28095606 0.77 KDM4E (0.55) S1PR1NR1H2NR1H3KDM4ETSHR
SCHEMBL28096010 0.77 KDM4E (0.55) S1PR1KDM4ETSHRPOLBHSD17B10
SCHEMBL28075492 0.77 KDM4E (0.62) S1PR1KDM4ETSHRPOLBHSD17B10
SCHEMBL28075481 0.76 KDM4E (0.57) S1PR1NR1H2NR1H3KDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN claimed
CN-106243130-B 3,6- diaryl-[1,2,4] triazole simultaneously [3,4-b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2019-03-01 CN disclosed
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN disclosed