SCHEMBL28095606

SCHEMBL28095606

COc1ccc(-c2n[nH]c(-c3cc(OC)c(OC)c(OC)c3)n2)cc1F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.55
POLB P06746 1/20 0.55
TSHR P16473 1/20 0.55
HSD17B10 Q99714 1/20 0.50
PSEN1 P49768 1/20 0.49
PSEN2 P49810 1/20 0.49
APH1B Q8WW43 1/20 0.49
NCSTN Q92542 1/20 0.49
APH1A Q96BI3 1/20 0.49
PSENEN Q9NZ42 1/20 0.49
S1PR1 P21453 1/20 0.46
ALDH1A1 P00352 3/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
NR1H2 P55055 1/20 0.45
NR1H3 Q13133 1/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
GRK6 P43250 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28096008 0.92 KDM4E (0.55) KDM4EPOLBTSHRHSD17B10PSEN1
SCHEMBL28833548 0.86 KDM4E (0.57) KDM4EPOLBTSHRHSD17B10PSEN1
SCHEMBL28095604 0.85 AMY1A (0.46) KDM4EHSD17B10PSEN1PSEN2APH1B
SCHEMBL28075492 0.84 KDM4E (0.62) KDM4EPOLBTSHRHSD17B10S1PR1
SCHEMBL28096010 0.84 KDM4E (0.55) KDM4EPOLBTSHRHSD17B10S1PR1
SCHEMBL17280055 0.83 KDM4E (0.60) KDM4EPOLBTSHRHSD17B10PSEN1
SCHEMBL28075488 0.82 KDM4E (0.58) KDM4EPOLBTSHRHSD17B10ALDH1A1
SCHEMBL28095619 0.81 KDM4E (0.57) KDM4EPOLBTSHRHSD17B10PSEN1
SCHEMBL17279690 0.81 NR1H2 (0.60) KDM4EPOLBTSHRALDH1A1MEN1
SCHEMBL6581499 0.80 NR1H2 (0.50) KDM4ETSHRHSD17B10PSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN claimed
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN disclosed