SCHEMBL28096012

SCHEMBL28096012

COc1ccc(-c2n[nH]c(-c3ccc(OC)c(OC)c3OC)n2)cc1OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.48
PDE4B Q07343 3/20 0.48
PDE4C Q08493 3/20 0.48
PDE4D Q08499 3/20 0.48
MAPT P10636 3/20 0.48
MAPK1 P28482 1/20 0.48
S1PR1 P21453 1/20 0.43
TSHR P16473 2/20 0.43
BRD4 O60885 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KDM4E B2RXH2 2/20 0.43
HSD17B10 Q99714 2/20 0.43
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
PSEN1 P49768 1/20 0.43
PSEN2 P49810 1/20 0.43
APH1B Q8WW43 1/20 0.43
NCSTN Q92542 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28096009 0.88 PDE4A (0.51) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL28096083 0.78 MAPT (0.49) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL28095604 0.78 AMY1A (0.46) MAPTS1PR1NPC1RAB9AKDM4E
SCHEMBL28075584 0.78 KDM4E (0.48) TSHRKDM4EHSD17B10ALDH1A1GAA
SCHEMBL28833481 0.78 AMY1A (0.46) MAPTNPC1RAB9AKDM4EHSD17B10
SCHEMBL28106648 0.77 AMY1A (0.43) S1PR1TSHRNPC1RAB9AKDM4E
SCHEMBL28106612 0.76 AMY1A (0.46) MAPTKDM4ENR1H2NR1H3
SCHEMBL28835288 0.76 ADORA2A (0.47) PDE4BMAPTTSHRNPC1RAB9A
SCHEMBL28106611 0.76 ATAD2 (0.56) MAPTTSHRNPC1RAB9AKDM4E
Hydrochloric Acid SCHEMBL6581075 0.75 ADORA2A (0.58) PDE4APDE4BPDE4CPDE4DMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN claimed
CN-106243130-B 3,6- diaryl-[1,2,4] triazole simultaneously [3,4-b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2019-03-01 CN disclosed
CN-106243130-A 3,6 diaryl [1,2,4] triazole also [3,4 b] [1,3,4] diazthines compound and application thereof 沈阳药科大学 2016-12-21 CN disclosed