SCHEMBL28096201

SCHEMBL28096201

Cc1ncc2c(C#C[Si](C)(C)C)c[nH]c2n1

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 4/20 0.38
PDK4 Q16654 2/20 0.36
AAK1 Q2M2I8 2/20 0.31
PDK1 Q15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31586107 0.79 LRRK2 (0.47) PDK2PDK4
SCHEMBL1796396 0.76 AAK1 (0.40) AAK1
SCHEMBL22525223 0.72 PDK2 (0.46) PDK2PDK4PDK1
SCHEMBL25304749 0.71 AURKA (0.46) AAK1
SCHEMBL19667381 0.69 PDK2 (0.44) PDK2PDK4PDK1
SCHEMBL19306614 0.69 PDK2 (0.49) PDK2PDK4PDK1
SCHEMBL5925906 0.68 LMNA (0.40)
SCHEMBL22883506 0.64 PDK2 (0.36) PDK2PDK4
SCHEMBL7842455 0.64 PARP1 (0.36)
SCHEMBL18874539 0.64 ALDH1A1 (0.40) PDK2PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106008512-B E1 activating enzyme inhibitors 千禧药品公司 2019-03-12 CN disclosed
CN-106008512-A INHIBITORS OF E1 ACTIVATING ENZYMES 千禧药品公司 2016-10-12 CN disclosed