SCHEMBL7842455

SCHEMBL7842455

Cc1nc2[nH]cc(C#C[Si](C)(C)C)c2c(=O)[nH]1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 5/20 0.36
TYMS P04818 8/20 0.35
MAPK1 P28482 1/20 0.33
TNKS2 Q9H2K2 1/20 0.31
CHUK O15111 1/20 0.31
CREBBP Q92793 1/20 0.30
CDK4 P11802 1/20 0.30
CCND1 P24385 1/20 0.30
ALDH1A1 P00352 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26232174 0.80 CHUK (0.49) CHUK
SCHEMBL7854494 0.74 TYMS (0.43) TYMS
SCHEMBL7851328 0.72 DAO (0.33) PARP1TYMSMAPK1ALDH1A1L3MBTL1
SCHEMBL7851196 0.71 TYMS (0.48) PARP1TYMSMAPK1TNKS2CDK4
SCHEMBL26232177 0.70 TYMS (0.41) PARP1TYMSMAPK1TNKS2ALDH1A1
SCHEMBL31022852 0.70 CHUK (0.44) CHUK
SCHEMBL4682893 0.65 GRIN2D (0.38) CREBBPALDH1A1
SCHEMBL5527750 0.65 RET (0.38) MAPK1CHUKALDH1A1
SCHEMBL1735020 0.64 CHEK1 (0.50) CHUK
SCHEMBL28096201 0.64 PDK2 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923287-A4 NONCLASSICAL PYRROLO 2,3-D]PYRIMIDINE ANTIFOLATES LILLY CO ELI (US) 2001-08-01 EP disclosed
EP-0923287-A1 NONCLASSICAL PYRROLO 2,3-D]PYRIMIDINE ANTIFOLATES ELI LILLY AND COMPANY (US) 1999-06-23 EP disclosed
WO-1998008382-A1 NONCLASSICAL PYRROLO[2,3-D]PYRIMIDINE ANTIFOLATES ELI LILLY AND COMPANY (US) 1998-03-05 WO disclosed