SCHEMBL28097694

SCHEMBL28097694

O=Cc1oc(-c2ccccc2)nc1O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.44
RAB9A P51151 5/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
MAPT P10636 4/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
KMT2A Q03164 1/20 0.43
IKBKB O14920 1/20 0.42
ELANE P08246 1/20 0.42
KDM4E B2RXH2 2/20 0.41
DHODH Q02127 1/20 0.40
GAA P10253 1/20 0.40
USP1 O94782 1/20 0.39
USP19 O94966 1/20 0.39
WDR48 Q8TAF3 1/20 0.39
PPARG P37231 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15265475 0.79 GAA (0.50) NPC1RAB9ASMN1; SMN2ALDH1A1IKBKB
SCHEMBL4852553 0.78 KDM4E (0.48) NPC1RAB9ASMN1; SMN2MAPTCYP1A2
SCHEMBL2364162 0.75 NPC1 (0.54) NPC1RAB9ASMN1; SMN2MAPTCYP1A2
SCHEMBL2903900 0.73 USP1 (0.47) NPC1RAB9ASMN1; SMN2MAPTCYP1A2
SCHEMBL27996878 0.73 GAA (0.55) NPC1RAB9ASMN1; SMN2MAPTCYP1A2
SCHEMBL5212183 0.72 FAAH (0.48) NPC1RAB9ASMN1; SMN2MAPTCYP1A2
SCHEMBL7738122 0.72 KDM4E (0.56) NPC1RAB9ASMN1; SMN2KDM4EGAA
SCHEMBL4029802 0.71 TSHR (0.38) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL5505905 0.69 USP1 (0.47) NPC1RAB9ASMN1; SMN2MAPTCYP1A2
SCHEMBL5638728 0.69 ESR2 (0.49) NPC1RAB9AMAPTALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106279132-B 2, 4-imidazoline diketone heterocyclic derivative and preparation method and application thereof 四川大学华西医院 2019-11-26 CN disclosed
CN-106279132-A 2, 4-imidazoline diketone heterocyclic derivative and preparation method and application thereof 四川大学华西医院 2017-01-04 CN disclosed