SCHEMBL28099847

SCHEMBL28099847

Cc1ccccc1N(C(N)=O)c1ccc(N)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
PLA2G7 Q13093 1/20 0.39
MAPK14 Q16539 2/20 0.38
MAPK13 O15264 1/20 0.38
MAPK12 P53778 1/20 0.38
MAPK11 Q15759 1/20 0.38
HSD17B10 Q99714 2/20 0.38
TSHR P16473 2/20 0.38
ALDH1A1 P00352 2/20 0.38
THRB P10828 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
CASP1 P29466 1/20 0.38
RECQL P46063 1/20 0.38
CHRM2 P08172 1/20 0.36
CHRM3 P20309 1/20 0.36
MAOA P21397 1/20 0.36
HTR2C P28335 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1954826 0.81 SIGMAR1 (0.44) CYP3A4TSHRALDH1A1HPGDMAPT
SCHEMBL28100008 0.81 CYP3A4 (0.50) CYP3A4CYP2C9CYP2C19HSD17B10TSHR
SCHEMBL28834470 0.80 KMT2A (0.48) CYP3A4CYP2C9CYP2C19HSD17B10TSHR
SCHEMBL6207117 0.80 CA2 (0.44) HSD17B10ALDH1A1HPGDHSD17B1HSD17B2
SCHEMBL7416227 0.77 SIGMAR1 (0.37) CYP3A4CYP2C9CYP2C19MAPK14MAPK13
SCHEMBL28099849 0.75 CYP3A4 (0.41) CYP3A4CYP2C9CYP2C19HSD17B10TSHR
SCHEMBL6256662 0.74 CES2 (0.41) MAPK14HSD17B10TSHRALDH1A1HTR3A
SCHEMBL6037570 0.74 TP53 (0.38) CYP2C19HSD17B10TSHRMAPTMEN1
SCHEMBL27455559 0.72 SIGMAR1 (0.38) CYP3A4TSHRALDH1A1HPGDHSD17B1
Hydrochloric Acid SCHEMBL9316439 0.72 SIGMAR1 (0.40) CYP3A4CYP2C9CYP2C19PLA2G7TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105884699-B 4- substituted aniline quinazoline derivative and its preparation method and application 中国药科大学 2019-05-07 CN disclosed
CN-105884699-A 4-substituted anilinoquinazoline derivatives, and preparation method and application thereof 中国药科大学 2016-08-24 CN disclosed