SCHEMBL28103993

SCHEMBL28103993

FC(F)(F)c1ccc2c(-c3ccccc3)cc(-c3ccccc3)nc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 4/20 0.57
ACACA Q13085 3/20 0.49
ESR1 P03372 1/20 0.47
NPBWR1 P48145 1/20 0.46
MET P08581 1/20 0.45
KDM4E B2RXH2 3/20 0.44
MAPK1 P28482 2/20 0.44
ALDH1A1 P00352 2/20 0.44
MAPT P10636 2/20 0.44
METAP2 P50579 1/20 0.44
MEN1 O00255 1/20 0.44
LMNA P02545 1/20 0.44
RECQL P46063 1/20 0.44
KMT2A Q03164 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
GRM4 Q14833 1/20 0.44
DGAT1 O75907 1/20 0.43
KCNH2 Q12809 1/20 0.43
ACP1 P24666 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28118653 0.89 TOP1 (0.58) TOP1ACACAESR1NPBWR1KDM4E
SCHEMBL25171878 0.88 TOP1 (0.68) TOP1ACACAKDM4EMAPK1ALDH1A1
SCHEMBL28046863 0.85 ESR1 (0.45) TOP1ESR1NPBWR1METKDM4E
SCHEMBL22983973 0.85 ACHE (0.64) TOP1ESR1NPBWR1METKDM4E
SCHEMBL5931070 0.81 TOP1 (0.60) TOP1ACACAMETKDM4EMAPK1
SCHEMBL13458752 0.80 TOP1 (0.59) TOP1ACACAMETKDM4EMAPT
SCHEMBL28170035 0.78 GRM4 (0.67) TOP1NPBWR1METGRM4KIF11
SCHEMBL1042853 0.77 ACACA (0.72) TOP1ACACAKDM4EMAPK1ALDH1A1
SCHEMBL29399315 0.77 ACACA (0.72) TOP1ACACAKDM4EMAPK1ALDH1A1
SCHEMBL5931163 0.77 TOP1 (0.49) TOP1METAP2KCNH2HPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106366035-B Synthesis method of quinoline derivative 南阳师范学院 2021-05-07 CN disclosed
CN-106380463-B Method for synthesizing quinoline derivative 南阳师范学院 2020-12-15 CN disclosed
CN-105175328-B It is a kind of using aromatic amine, aromatic aldehyde, ketone synthesis of quinoline derivatives method 南阳师范学院 2017-12-19 CN disclosed
CN-106380463-A Method for synthesis of quinoline derivatives 南阳师范学院 2017-02-08 CN disclosed
CN-106366035-A Method for synthesizing quinoline derivative 南阳师范学院 2017-02-01 CN disclosed