SCHEMBL28106567

SCHEMBL28106567

COC(=O)c1ccc(Oc2ccc(Oc3ccccc3)cc2)nc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.61
ALDH1A1 P00352 1/20 0.55
GAA P10253 1/20 0.55
MAPT P10636 1/20 0.55
RAB9A P51151 1/20 0.55
OPRM1 P35372 7/20 0.54
OPRD1 P41143 7/20 0.54
OPRK1 P41145 5/20 0.54
GRN P28799 2/20 0.53
SORT1 Q99523 2/20 0.53
MAPK1 P28482 2/20 0.53
KDM4E B2RXH2 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
HRH3 Q9Y5N1 1/20 0.52
CTSA P10619 1/20 0.50
GRIN2D O15399 1/20 0.49
GRIN3B O60391 1/20 0.49
SLC6A2 P23975 1/20 0.49
SLC6A3 Q01959 1/20 0.49
GRIN1 Q05586 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3586183 0.97 LMNA (0.60) LMNAALDH1A1GAAMAPTRAB9A
SCHEMBL6339006 0.87 OPRM1 (0.57) LMNAMAPTRAB9AOPRM1OPRD1
SCHEMBL21656526 0.87 LMNA (0.63) LMNAALDH1A1GAARAB9AMAPK1
SCHEMBL12157057 0.85 LMNA (0.65) LMNAALDH1A1MAPK1KDM4EL3MBTL1
SCHEMBL15684885 0.85 LMNA (0.61) LMNAALDH1A1MAPTRAB9AMAPK1
SCHEMBL619879 0.85 LMNA (0.61) LMNAALDH1A1MAPTRAB9AOPRM1
SCHEMBL21656974 0.84 LMNA (0.60) LMNAMAPTRAB9AOPRM1OPRD1
SCHEMBL31646829 0.83 L3MBTL1 (0.54) LMNAALDH1A1GAAMAPTMAPK1
SCHEMBL21656686 0.83 LMNA (0.59) LMNAALDH1A1OPRM1OPRD1MAPK1
SCHEMBL29596790 0.83 RXFP1 (0.56) ALDH1A1GAAMAPTRAB9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105939998-A Heteroaryl compounds as btk inhibitors and uses thereof 默克专利有限公司 2016-09-14 CN disclosed