SCHEMBL28107195

SCHEMBL28107195

N#Cc1c[nH]c2cc(-c3cccnc3)ccc12

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 1/20 0.57
CDK9 P50750 1/20 0.57
HASPIN Q8TF76 1/20 0.57
CYP11B2 P19099 2/20 0.49
TDO2 P48775 2/20 0.49
QPCT Q16769 1/20 0.49
QPCTL Q9NXS2 1/20 0.49
CYP17A1 P05093 1/20 0.49
CYP11B1 P15538 1/20 0.49
IMPDH2 P12268 2/20 0.47
IMPDH1 P20839 1/20 0.47
FGFR1 P11362 1/20 0.47
LRRK2 Q5S007 1/20 0.47
FLT3 P36888 2/20 0.46
NR4A2 P43354 1/20 0.45
GSK3B P49841 1/20 0.44
DYRK1A Q13627 1/20 0.44
NEK1 Q96PY6 1/20 0.44
CHEK1 O14757 2/20 0.43
FASN P49327 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29957979 0.75 CCNT1 (0.57) CCNT1CDK9HASPINTDO2QPCT
SCHEMBL22482294 0.74 CCNT1 (0.62) CCNT1CDK9HASPINIMPDH2IMPDH1
SCHEMBL3319584 0.72 CYP11B2 (0.56) CYP11B2CYP17A1CYP11B1FASN
SCHEMBL6773157 0.72 CYP11B2 (0.56) CYP11B2CYP17A1CYP11B1
SCHEMBL6439562 0.72 CYP11B2 (0.56) CYP11B2CYP17A1CYP11B1
SCHEMBL19128281 0.72 CYP11B2 (0.70) CYP11B2CYP17A1CYP11B1
SCHEMBL10707057 0.71 PIK3CD (0.68) CYP11B2CYP17A1CYP11B1FASN
SCHEMBL31663544 0.71 XDH (0.55) CYP11B2CYP17A1CYP11B1
SCHEMBL15667411 0.71 CCNT1 (0.62) CCNT1CDK9HASPINIMPDH2IMPDH1
SCHEMBL11653917 0.70 NR4A2 (0.58) HASPINTDO2QPCTQPCTLNR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104193725-B Organic compound 诺华股份有限公司 2016-11-16 CN disclosed