SCHEMBL28110445

SCHEMBL28110445

c1ccc2c(c1)CCN=C2CN1CCOCC1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.56
KDM4E B2RXH2 1/20 0.56
NPC1 O15118 1/20 0.49
TP53 P04637 1/20 0.49
TSHR P16473 1/20 0.49
MAPK1 P28482 1/20 0.49
RAB9A P51151 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
CXCR4 P61073 1/20 0.45
NOS3 P29474 1/20 0.44
NOS2 P35228 1/20 0.44
CYP2A13 Q16696 5/20 0.43
PTAFR P25105 1/20 0.42
USP2 O75604 1/20 0.42
CYP3A4 P08684 1/20 0.42
THRB P10828 1/20 0.42
MAPT P10636 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3451869 0.86 ALDH1A1 (0.60) ALDH1A1KDM4ENOS3NOS2PTAFR
SCHEMBL7699664 0.78 HRH3 (0.55) ALDH1A1NPC1TP53TSHRMAPK1
SCHEMBL7706897 0.73 ALDH1A1 (0.50) ALDH1A1NPC1TP53TSHRMAPK1
SCHEMBL7698346 0.73 TSHR (0.42) ALDH1A1NPC1TP53TSHRMAPK1
SCHEMBL29361631 0.73 KDM4E (0.60) ALDH1A1KDM4ETP53MEN1KMT2A
SCHEMBL7509399 0.73 KDM4E (0.60) ALDH1A1KDM4ETP53MEN1KMT2A
SCHEMBL7703268 0.73 CYP2A13 (0.41) ALDH1A1NPC1TP53TSHRMAPK1
SCHEMBL7701109 0.73 TSHR (0.41) ALDH1A1NPC1TP53TSHRMAPK1
SCHEMBL14919523 0.72 ALDH1A1 (1.00) ALDH1A1KDM4ENPC1TSHRRAB9A
SCHEMBL30952110 0.72 ALDH1A1 (1.00) ALDH1A1KDM4ENPC1TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105431422-B Isoindoline or isoquinoline compounds, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2019-08-30 CN disclosed
CN-109456324-A New isoindoline or isoquinoline compound, preparation method and the Pharmaceutical composition containing them 法国施维雅药厂 2019-03-12 CN disclosed
CN-105408321-B Indoles and azole derivatives, their preparation method and the pharmaceutical composition containing them 法国施维雅药厂 2019-03-08 CN disclosed
CN-104341451-B New phosphate compound, its preparation method and the pharmaceutical composition containing them 瑟维尔实验室 2018-04-03 CN disclosed
CN-104341395-B Novel azole compounds, process for their preparation and pharmaceutical compositions containing them 瑟维尔实验室 2017-07-04 CN disclosed
CN-106674201-A Pyrrole compounds, method of preparing same and pharmaceutical compositions containing the compounds 法国施维雅药厂 2017-05-17 CN disclosed
CN-106674196-A Pyrrole compounds, method of preparing same and pharmaceutical compositions containing them 法国施维雅药厂 2017-05-17 CN disclosed
CN-104144930-B New indolizine derivatives, method for preparing same and pharmaceutical compositions containing same 瑟维尔实验室 2017-02-22 CN disclosed