SCHEMBL7706897

SCHEMBL7706897

Cn1cc(CN2CCOCC2)c(C2=NCCc3ccccc32)n1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.50
KMT2A Q03164 3/20 0.50
POLB P06746 2/20 0.50
LMNA P02545 1/20 0.50
CYP2A13 Q16696 3/20 0.45
MEN1 O00255 2/20 0.43
DRD4 P21917 1/20 0.43
PLA2G7 Q13093 1/20 0.43
MGLL Q99685 1/20 0.43
ABHD6 Q9BV23 1/20 0.43
MAPT P10636 2/20 0.42
NPC1 O15118 2/20 0.41
ATM Q13315 1/20 0.40
SLC2A1 P11166 1/20 0.40
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7703268 0.79 CYP2A13 (0.41) ALDH1A1KMT2ALMNACYP2A13MEN1
SCHEMBL7698346 0.77 TSHR (0.42) ALDH1A1KMT2APOLBLMNACYP2A13
SCHEMBL7699664 0.77 HRH3 (0.55) ALDH1A1KMT2ALMNACYP2A13MEN1
SCHEMBL7701109 0.76 TSHR (0.41) ALDH1A1KMT2ALMNACYP2A13MEN1
SCHEMBL28110445 0.73 ALDH1A1 (0.56) ALDH1A1KMT2ALMNACYP2A13MEN1
SCHEMBL8510483 0.71 CYP2A13 (0.40) ALDH1A1KMT2APOLBLMNACYP2A13
SCHEMBL15266951 0.70 PLA2G7 (0.56) ALDH1A1KMT2ALMNAMEN1PLA2G7
SCHEMBL7699631 0.69 CHKA (0.53) LMNANPC1TP53RAB9A
SCHEMBL7702406 0.68 OPRM1 (0.41) ALDH1A1KMT2APOLBLMNACYP2A13
SCHEMBL7702411 0.68 OPRM1 (0.41) ALDH1A1KMT2APOLBLMNACYP2A13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1098260-C 2,4-diaminopyrimidine derivatives BASLIR PHARMACEUTICALS AG (CH) 2003-01-08 CN disclosed
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
CN-1218465-A 2,4-diaminopyrimidine derivatives HOFFMANN LA ROCHE (CH) 1999-06-02 CN disclosed
EP-0901488-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-03-17 EP disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed
WO-1997043277-A1 2,4-DIAMINOPYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1997-11-20 WO disclosed