SCHEMBL7698346

SCHEMBL7698346

Cn1nc(CN2CCOCC2)cc1C1=NCCc2ccccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CXCR4 P61073 1/20 0.41
KCNH2 Q12809 1/20 0.41
USP2 O75604 1/20 0.39
CYP3A4 P08684 1/20 0.39
THRB P10828 1/20 0.39
MAPT P10636 2/20 0.37
LMNA P02545 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GAA P10253 1/20 0.37
CYP2A13 Q16696 2/20 0.36
ALDH1A1 P00352 3/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7701109 0.81 TSHR (0.41) TSHRNPC1TP53MAPK1RAB9A
SCHEMBL7706897 0.77 ALDH1A1 (0.50) TSHRNPC1TP53MAPK1RAB9A
SCHEMBL7705891 0.77 ALDH1A1 (0.38) LMNAALDH1A1
SCHEMBL7702368 0.76 NOS3 (0.41) SMN1; SMN2KCNH2MAPTLMNAALDH1A1
SCHEMBL7703268 0.76 CYP2A13 (0.41) TSHRNPC1TP53MAPK1RAB9A
SCHEMBL7700170 0.76 NOS3 (0.38) MAPTLMNAALDH1A1KMT2AMEN1
SCHEMBL7699664 0.75 HRH3 (0.55) TSHRNPC1TP53MAPK1RAB9A
SCHEMBL28110445 0.73 ALDH1A1 (0.56) TSHRNPC1TP53MAPK1RAB9A
SCHEMBL7703215 0.71 KMT2A (0.44) ALDH1A1KMT2AMEN1POLB
SCHEMBL8509692 0.71 CXCR4 (0.39) TSHRNPC1TP53MAPK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1098260-C 2,4-diaminopyrimidine derivatives BASLIR PHARMACEUTICALS AG (CH) 2003-01-08 CN disclosed
EP-0901488-B1 2,4-DIAMINOPYRIMIDINE DERIVATIVES BASILEA PHARMACEUTICA AG (CH) 2002-11-06 EP disclosed
CN-1218465-A 2,4-diaminopyrimidine derivatives HOFFMANN LA ROCHE (CH) 1999-06-02 CN disclosed
US-5866583-A Substituted 2,4-diaminopyrimidines HOFFMANN-LA ROCHE INC. (US) 1999-02-02 US disclosed