SCHEMBL28110995

SCHEMBL28110995

C=CC(=O)N1CCCC(C#N)C1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 11/20 0.41
EGFR P00533 3/20 0.39
BTK Q06187 2/20 0.38
JAK1 P23458 1/20 0.38
VNN1 O95497 3/20 0.37
BTD P43251 2/20 0.37
DPP4 P27487 2/20 0.37
MAP2K7 O14733 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23221969 0.83 EGFR (0.41) JAK3EGFRBTKJAK1MAP2K7
SCHEMBL18173568 0.79 JAK3 (0.44) JAK3EGFRBTKJAK1MAP2K7
SCHEMBL18173596 0.79 JAK3 (0.44) JAK3EGFRBTKJAK1MAP2K7
SCHEMBL28168621 0.79 VNN1 (0.40) VNN1BTDDPP4
SCHEMBL20456230 0.79 TEAD1 (0.39) JAK3BTKJAK1DPP4
SCHEMBL18478125 0.77 ALDH1A1 (0.40) VNN1BTDDPP4
SCHEMBL18478943 0.77 ALDH1A1 (0.40) VNN1BTDDPP4
SCHEMBL30208798 0.75 CA12 (0.47) JAK3EGFRBTKJAK1
SCHEMBL8362428 0.75 CA12 (0.47) JAK3EGFRBTKJAK1
SCHEMBL16802109 0.75 CA12 (0.47) JAK3EGFRBTKJAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106061973-B Pyrrolo [2,3-D ] pyrimidinyl, pyrrolo [2,3-B ] pyrazinyl and pyrrolo [2,3-D ] pyridylacrylamide 辉瑞公司 2019-07-09 CN disclosed
CN-107417684-A Heterocyclic acryloyloxy amine 辉瑞公司 2017-12-01 CN disclosed
CN-106061973-A Pyrrolo [2,3-D ] pyrimidinyl, pyrrolo [2,3-B ] pyrazinyl and pyrrolo [2,3-D ] pyridylacrylamide 辉瑞公司 2016-10-26 CN disclosed