SCHEMBL28111052

SCHEMBL28111052

O=C(O)c1cc(OCC(F)(F)F)[nH]n1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 15/20 0.45
DAO P14920 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
HCAR3 P49019 3/20 0.40
CYTH3 O43739 1/20 0.40
BTK Q06187 1/20 0.40
EPN1 Q9Y6I3 1/20 0.40
ASPH Q12797 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31068051 0.86 KMT2A (0.38) L3MBTL1
SCHEMBL17224847 0.83 MAPK1 (0.51) HCAR2L3MBTL1
SCHEMBL15467909 0.78 HCAR2 (0.56) HCAR2DAOHCAR3CYTH3BTK
SCHEMBL28015264 0.74 L3MBTL1 (0.49) HCAR2L3MBTL1HCAR3ASPH
SCHEMBL28488240 0.74 HCAR2 (0.43) HCAR2DAOHCAR3CYTH3BTK
SCHEMBL16445300 0.74 HCAR2 (0.60) HCAR2DAOHCAR3CYTH3BTK
SCHEMBL219145 0.73 ALDH1A1 (0.44) L3MBTL1
SCHEMBL5317023 0.72 HCAR2 (0.58) HCAR2DAOHCAR3CYTH3BTK
SCHEMBL2360520 0.72 HCAR2 (0.52) HCAR2DAOHCAR3CYTH3BTK
SCHEMBL15350209 0.70 CNR2 (0.42) HCAR2DAOL3MBTL1ASPH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106255688-B Morpholine-pyridine derivate 豪夫迈·罗氏有限公司 2019-11-08 CN disclosed
CN-106255688-A Morpholine pyridine derivate 豪夫迈·罗氏有限公司 2016-12-21 CN disclosed