SCHEMBL28111553

SCHEMBL28111553

COC(=O)c1cn(Br)c2ncc(Br)nc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.37
POLB P06746 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
KDM4E B2RXH2 7/20 0.36
ALDH1A1 P00352 5/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
KMT2A Q03164 5/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
HPGD P15428 2/20 0.33
OPRK1 P41145 2/20 0.33
HSD17B10 Q99714 2/20 0.33
MEN1 O00255 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
CYP2C9 P11712 1/20 0.33
TSHR P16473 1/20 0.33
PDE1B Q01064 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14737356 0.78 ABCB11 (0.33) LMNAPOLBTDP1KDM4EALDH1A1
SCHEMBL1372546 0.77 DGAT1 (0.41) LMNAPOLBTDP1KDM4EALDH1A1
SCHEMBL14737300 0.76 LMNA (0.38) LMNAPOLBTDP1KDM4EALDH1A1
SCHEMBL14737585 0.71 MAPK1 (0.51) CYP2C9MAPK1
SCHEMBL31153593 0.67 NR4A2 (0.50) LMNAKDM4EALDH1A1KMT2AL3MBTL1
SCHEMBL30570809 0.66 NPSR1 (0.56) KDM4EALDH1A1L3MBTL1MAPK1
SCHEMBL14751302 0.66 SYK (0.39) LMNA
SCHEMBL18534427 0.65 JAK3 (0.34) POLBALDH1A1KMT2AMEN1CYP2C9
SCHEMBL29411823 0.65 NPSR1 (0.48) KDM4EALDH1A1L3MBTL1TSHRMAPK1
SCHEMBL30050535 0.65 ATR (0.54) KDM4EALDH1A1L3MBTL1SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106061973-A Pyrrolo [2,3-D ] pyrimidinyl, pyrrolo [2,3-B ] pyrazinyl and pyrrolo [2,3-D ] pyridylacrylamide 辉瑞公司 2016-10-26 CN disclosed