SCHEMBL28111580

SCHEMBL28111580

Nc1nc2cc[nH]c2nc1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 4/20 0.40
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAPK8 P45983 1/20 0.32
MAPK9 P45984 1/20 0.32
MAPK10 P53779 1/20 0.32
TTK P33981 1/20 0.32
JAK2 O60674 1/20 0.31
AXL P30530 1/20 0.31
CDK8 P49336 1/20 0.31
APP P05067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25934515 0.73 MAPK1 (0.50) MAPK1KDM4EALDH1A1GAAMAPT
SCHEMBL28111579 0.69 TTK (0.39) MAPK8TTKJAK2CDK8
SCHEMBL977078 0.66 CSNK1A1 (0.48) MAPK1
SCHEMBL29870187 0.66 CSNK1A1 (0.48) MAPK1
SCHEMBL4559275 0.66 MAPT (0.52) MAPK1KDM4EALDH1A1GAAMAPT
SCHEMBL14104385 0.65 MAPK1 (0.41) MAPK1AXL
SCHEMBL25934516 0.64 MAPK1 (0.44) MAPK1
SCHEMBL16415962 0.62 HTR6 (0.53) MAPK1KDM4EALDH1A1GAAMAPT
SCHEMBL20209150 0.62 MAPK1 (0.40) MAPK1
SCHEMBL20208921 0.62 ALDH1A1 (0.41) MAPK1ALDH1A1MAPTJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106061973-A Pyrrolo [2,3-D ] pyrimidinyl, pyrrolo [2,3-B ] pyrazinyl and pyrrolo [2,3-D ] pyridylacrylamide 辉瑞公司 2016-10-26 CN disclosed