SCHEMBL28113418

SCHEMBL28113418

O=c1ccccn1-n1cccn1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.38
CA1 P00915 3/20 0.38
CA2 P00918 3/20 0.38
CA9 Q16790 3/20 0.38
ADORA3 P0DMS8 1/20 0.36
CA14 Q9ULX7 1/20 0.34
PDE4B Q07343 2/20 0.33
TSHR P16473 1/20 0.33
ELANE P08246 2/20 0.32
POLB P06746 2/20 0.32
PKM P14618 1/20 0.32
MAPK1 P28482 2/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
NPC1 O15118 1/20 0.31
CHRM1 P11229 1/20 0.31
GAA P10253 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1191487 0.75 MEN1 (0.40) CA12CA1CA2CA9ADORA3
SCHEMBL3985923 0.74 KDM4E (0.33) KDM4EALDH1A1
SCHEMBL18284673 0.74 CYP19A1 (0.39) CA12CA1CA2CA9ADORA3
SCHEMBL31740751 0.73 CA12 (0.39) CA12CA1CA2CA9MAPK1
SCHEMBL28099160 0.69 POLB (0.44) CA12CA1CA2CA9ADORA3
SCHEMBL9464929 0.67 NOS1 (0.38) MAPK1KDM4EALDH1A1NPC1GAA
SCHEMBL27816541 0.66 CA12 (0.44) CA12CA9TSHRMAPK1ALDH1A1
SCHEMBL7627710 0.64 POLB (0.35) CA12CA1CA2CA9ADORA3
SCHEMBL30415564 0.63 RECQL (0.38) CA12CA1CA2CA9CA14
SCHEMBL1205563 0.63

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106170489-B New Pyrazolopyrimidine derivative and its purposes as MALT1 inhibitor 诺华股份有限公司 2019-05-03 CN disclosed
CN-106170489-A New Pyrazolopyrimidine derivative and the purposes as MALT1 inhibitor thereof 诺华股份有限公司 2016-11-30 CN disclosed