SCHEMBL28113638

SCHEMBL28113638

COc1cccc(-c2n[nH]cc2N)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 4/20 0.50
GAA P10253 1/20 0.50
PIK3CG P48736 1/20 0.49
DCUN1D1 Q96GG9 1/20 0.49
ADORA1 P30542 3/20 0.48
TP53 P04637 1/20 0.48
HPGD P15428 1/20 0.48
HTT P42858 1/20 0.48
ADORA2B P29275 1/20 0.48
KDM4E B2RXH2 1/20 0.48
KMT2A Q03164 1/20 0.48
DYRK1A Q13627 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
DPP4 P27487 1/20 0.47
TDO2 P48775 1/20 0.47
ALDH1A1 P00352 2/20 0.46
CYP3A4 P08684 1/20 0.46
NOTUM Q6P988 1/20 0.46
NR1H2 P55055 1/20 0.46
NR1H3 Q13133 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17895374 0.81 GAA (0.50) ADORA2AGAADCUN1D1ADORA1TP53
SCHEMBL29484271 0.81 GAA (0.50) ADORA2AGAADCUN1D1ADORA1TP53
SCHEMBL2314103 0.80 RAB9A (0.46) PIK3CGADORA1TP53HPGDKMT2A
SCHEMBL4700185 0.79 TDO2 (0.55) ADORA2APIK3CGADORA1KDM4EKMT2A
SCHEMBL942446 0.77 ADORA2A (0.46) ADORA2AADORA1ADORA2BDPP4TDO2
SCHEMBL28113133 0.77 PIK3CG (0.47) ADORA2APIK3CGADORA1ADORA2BDYRK1A
SCHEMBL2379590 0.75 ALOX15 (0.48) ADORA2AGAAADORA1HPGDKDM4E
SCHEMBL544500 0.75 ALOX15 (0.48) ADORA2AGAAADORA1HPGDKDM4E
SCHEMBL27866855 0.74 DYRK1A (0.60) ADORA2APIK3CGADORA1TP53HPGD
SCHEMBL15428616 0.73 ADORA2A (0.51) ADORA2APIK3CGADORA1ADORA2BCLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106188059-A Some chemical entities, compositions and method 英特利凯恩有限责任公司 2016-12-07 CN disclosed