SCHEMBL28113661

SCHEMBL28113661

O=C(OC(=O)c1ccccn1)c1ccncc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.51
MAPT P10636 2/20 0.51
POLB P06746 1/20 0.51
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
NPC1 O15118 5/20 0.49
RAB9A P51151 5/20 0.49
KMT2A Q03164 4/20 0.49
PKM P14618 4/20 0.49
GAA P10253 2/20 0.49
CDK5 Q00535 2/20 0.49
CDK5R1 Q15078 2/20 0.49
MITF O75030 1/20 0.49
L3MBTL1 Q9Y468 4/20 0.48
LMNA P02545 2/20 0.48
NAPRT Q6XQN6 1/20 0.48
P4HTM Q9NXG6 1/20 0.48
ALDH1A1 P00352 1/20 0.47
HSD17B10 Q99714 1/20 0.46
PAX8 Q06710 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27454868 0.89 KMT2A (0.61) KDM4EMAPTPOLBCES2CES1
SCHEMBL31633615 0.87 CES2 (0.64) KDM4EMAPTPOLBCES2CES1
SCHEMBL1228223 0.87 CES2 (0.64) KDM4EMAPTPOLBCES2CES1
SCHEMBL31390431 0.86 CES2 (0.53) KDM4EMAPTPOLBCES2CES1
SCHEMBL11665942 0.81 KMT2A (0.65) MAPTPOLBNPC1RAB9AKMT2A
SCHEMBL647632 0.81 HSD17B10 (0.64) KDM4EPOLBNPC1RAB9AKMT2A
SCHEMBL8345410 0.79 CES2 (0.50) KDM4EMAPTPOLBCES2CES1
SCHEMBL16460100 0.78 KMT2A (0.78) KDM4EMAPTCES2CES1NPC1
SCHEMBL27505714 0.78 L3MBTL1 (0.61) KDM4EMAPTPOLBCES2CES1
SCHEMBL31135050 0.78 KMT2A (0.78) KDM4EMAPTCES2CES1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106491593-A The application of alantolactone derivant and its salt in treatment inflammatory bowel medicine is prepared 天承南运(天津)科技有限公司 2017-03-15 CN claimed
CN-106491592-A The application of alantolactone derivant and its salt in treatment thyroiditiss medicine is prepared 南开大学 2017-03-15 CN claimed
CN-106496243-A The application of isoalantolactone derivant and its salt in treatment pulmonary fibrosis medicine is prepared 南开大学 2017-03-15 CN claimed
CN-106491594-A The application of alantolactone derivant and its salt in treatment pulmonary fibrosis medicine is prepared 南开大学 2017-03-15 CN claimed
CN-106474109-A The application in preparation treatment inflammatory bowel medicine of isoalantolactone derivant and its salt 天承南运(天津)科技有限公司 2017-03-08 CN claimed