SCHEMBL28113776

SCHEMBL28113776

Cc1cccc(N(C)C)c1[N+](=O)[O-]

nearest known ligand 0.67

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.67
TDP1 Q9NUW8 3/20 0.67
TSHR P16473 4/20 0.58
SMN1; SMN2 Q16637 2/20 0.46
MAPT P10636 4/20 0.45
HSD17B10 Q99714 1/20 0.44
KAT2B Q92831 1/20 0.42
CYP3A4 P08684 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA4 P22748 1/20 0.39
CA9 Q16790 1/20 0.39
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2056581 0.83 TDP1 (0.64) ALDH1A1TDP1TSHRSMN1; SMN2MAPT
SCHEMBL635089 0.81 ALDH1A1 (1.00) ALDH1A1TDP1TSHRSMN1; SMN2MAPT
SCHEMBL6316759 0.80 ALDH1A1 (0.60) ALDH1A1TDP1TSHRSMN1; SMN2MAPT
SCHEMBL27363125 0.79 MAPT (0.44) ALDH1A1TDP1TSHRSMN1; SMN2MAPT
SCHEMBL30870615 0.79 MAPT (0.44) ALDH1A1TDP1TSHRSMN1; SMN2MAPT
SCHEMBL21543104 0.79 MAPT (0.44) ALDH1A1TDP1TSHRSMN1; SMN2MAPT
SCHEMBL8917458 0.79 MAPT (0.44) ALDH1A1TDP1TSHRMAPTCA12
SCHEMBL28521563 0.79 ALDH1A1 (0.95) ALDH1A1TDP1TSHRSMN1; SMN2MAPT
SCHEMBL10193193 0.78 TDP1 (0.50) ALDH1A1TDP1TSHRMAPTPOLB
SCHEMBL2566822 0.78 ALDH1A1 (0.56) ALDH1A1TDP1TSHRSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111718332-B 2-substituted pyrazol amino-4-substituted amino-5-pyrimidine formamide compound, composition and application thereof 北京赛特明强医药科技有限公司 2021-08-17 CN disclosed
CN-111718332-A 2-substituted pyrazol amino-4-substituted amino-5-pyrimidine formamide compound, composition and application thereof 北京赛特明强医药科技有限公司 2020-09-29 CN disclosed
CN-104487433-B Triazolone compounds as mPGES-1 inhibitors 格兰马克药品股份有限公司 2016-12-07 CN disclosed