SCHEMBL28114366

SCHEMBL28114366

OC1(c2ccccc2)C=CC=C(Br)C1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC9 Q9UKV0 1/20 0.39
HDAC4 P56524 3/20 0.33
HSD11B1 P28845 1/20 0.33
MAOB P27338 5/20 0.32
MAOA P21397 4/20 0.32
AKR1C1 Q04828 1/20 0.32
KDM4E B2RXH2 2/20 0.32
LMNA P02545 2/20 0.32
GAA P10253 2/20 0.32
MAPT P10636 2/20 0.32
MEN1 O00255 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL123293 0.79 MAOB (0.33) HDAC9MAOBMAOA
SCHEMBL28450776 0.78 CHRNB2 (0.36) HDAC9MAOBMAOAKDM4EGAA
SCHEMBL30559625 0.77 MEN1 (0.36) HDAC4LMNAMAPTMEN1KMT2A
SCHEMBL29044791 0.77 MEN1 (0.36) HDAC4LMNAMAPTMEN1KMT2A
SCHEMBL27897540 0.76 HDAC1 (0.41) HDAC9HDAC4MAOBMAOAALDH1A1
SCHEMBL17866314 0.76 HDAC9 (0.36) HDAC9HDAC4HSD11B1MEN1KMT2A
SCHEMBL28479583 0.69 RAB9A (0.38) HDAC9MAOA
SCHEMBL4942855 0.67 OPRL1 (0.35)
SCHEMBL29025928 0.67
SCHEMBL4089733 0.67 HDAC4 (0.36) HDAC9HDAC4MAOBMAOAAKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106117203-B A kind of synthetic method of 3 arylthio Imidazoheterocyclic compounds 安徽理工大学 2017-11-07 CN disclosed
CN-106117203-A A kind of synthetic method of 3 arylthio Imidazoheterocyclic compounds 安徽理工大学 2016-11-16 CN disclosed