SCHEMBL28114800

SCHEMBL28114800

COC(=O)c1ccc2c(ccn2Cl)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.48
ALDH1A1 P00352 5/20 0.48
HPGD P15428 4/20 0.48
HSD17B10 Q99714 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
POLB P06746 1/20 0.48
APOBEC3A P31941 1/20 0.48
APOBEC3G Q9HC16 1/20 0.48
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
CA12 O43570 2/20 0.46
CA7 P43166 2/20 0.46
CA9 Q16790 2/20 0.46
CA14 Q9ULX7 2/20 0.46
XDH P47989 1/20 0.46
LCK P06239 1/20 0.45
ALOX15 P16050 2/20 0.44
HTT P42858 2/20 0.44
PTPN11 Q06124 1/20 0.44
HDAC8 Q9BY41 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22489748 0.90 KDM4E (0.54) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL29944244 0.82 TUBB4A (0.59) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL108632 0.82 TUBB4A (0.59) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL13699049 0.81 KDM4E (0.55) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL28837051 0.81 CA1 (0.46) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL15822845 0.80 RAPGEF4 (0.48) KDM4EHSD17B10POLBCA1CA2
SCHEMBL18555462 0.79 KDM4E (0.48) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL26440951 0.78 KDM4E (0.44) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL2324058 0.78 TUBB4A (0.62) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2
SCHEMBL7880047 0.78 KDM4E (0.49) KDM4EALDH1A1HPGDHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109963849-A nitrogen-containing heterocyclic compounds as FXR modulators 合帕吉恩治疗公司 2019-07-02 CN disclosed
CN-107531679-A Aromatic amides analog derivative, its preparation method and its application in medicine 江苏恒瑞医药股份有限公司 2018-01-02 CN disclosed
CN-104812749-B Indolecarboxamide derivant as P2X7 receptor antagonist 埃科特莱茵药品有限公司 2016-12-14 CN disclosed